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Report error Found 8 of ec50 for UniProtKB: Q9Y271
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50292408(5S-hydroxy-6R-(S-cysteinylglycinyl)-7E,9E,11E,14Z-...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50596196(CHEBI:16978 | CHEMBL451509)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50052024(montelukast | CHEMBL787)
Affinity DataEC50:  72nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50297387((5S-(5R*,6S*(S*),7E,9E,11Z,14Z))-6-((2-Amino-2-car...)
Affinity DataEC50:  104nMAssay Description:Agonist activity at human CysLT1 receptorMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50323903((E)-4-(3-(4-(4-(4-Chlorophenoxy)butoxy)phenyl)acry...)
Affinity DataEC50:  480nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50323902((E)-2-(2-(3-(4-(4-(4-Chlorophenoxy)butoxy)phenyl)a...)
Affinity DataEC50:  1.30E+3nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50323901(E-2-(2-(3-(4-(4-(4-Chlorophenoxy)butoxy)phenyl)acr...)
Affinity DataEC50:  1.40E+3nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteinyl leukotriene receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50323904((E)-4-(Cyanomethoxy)-3-(3-(4-(4-phenoxybutoxy)phen...)
Affinity DataEC50:  3.90E+3nMAssay Description:Antagonist activity at CysLT1 receptor in human dU937 cells assessed as inhibition of LTD4-induced increase of calcium level treated 30 mins before L...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed