Compile Data Set for Download or QSAR
maximum 50k data
Found 188 of ki for UniProtKB: A0A480I924
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50292408((R-(R*,S*-(E,E,Z,Z)))-N-(S-(1-(4-Carboxy-1-hydroxy...)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50297387((5S,6R,7E,9E,11Z,14Z)-6-(cystein-S-yl)-5-hydroxyic...)
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM81801(CAS_5283121 | LTC4 | NSC_5283121)
Affinity DataKi:  3.58nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023962(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-hex-2...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023979(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-(3...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024024(2-[(2,2-Dibromo-cyclopropanecarbonyl)-amino]-but-2...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023951(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  40nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024072(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-et...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023999(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024019(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  58nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367508(CHEMBL1907817)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024071(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-oct-...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367506(CHEMBL1907823)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023983(2-[(2,2-Dichloro-cyclopropanecarbonyl)-amino]-but-...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023933(8-Cyano-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  82nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024023(CHEMBL276215 | Sodium; 6-carboxy-6-[(2,2-dimethyl-...)
Affinity DataKi:  87nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024055(2-{6-Carboxy-6-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023947(2,11-Bis-[(2,2-dimethyl-cyclopropanecarbonyl)-amin...)
Affinity DataKi:  92nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024044(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dec-...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023992(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-ph...)
Affinity DataKi:  100nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367502(CILASTATIN)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024045(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023942(10-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-am...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023995(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-dode...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023990(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hept...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024042(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-unde...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024036(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-5-me...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024069(7-Carboxymethylsulfanyl-2-[(2,2-dimethyl-cycloprop...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024003(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-(3...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024078(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-trid...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023971(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-hex-...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024059(7-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024012(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367507(CHEMBL1237318)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367505(CHEMBL1907816)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023963(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-6-me...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023946(4-Cyclohexyl-2-[(2,2-dimethyl-cyclopropanecarbonyl...)
Affinity DataKi:  150nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024066(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-non-...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024058(7-(2-Carboxy-2-oxo-ethylsulfanyl)-2-[(2,2-dimethyl...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367509(CHEMBL1907822)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024053(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-7-me...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024005(9-Bromo-2-[(2,2-dimethyl-cyclopropanecarbonyl)-ami...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023976((R)-2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023972(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023997(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-pent...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024008(CHEMBL11674 | {7-Carboxy-7-[(2,2-dichloro-cyclopro...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50367503(CHEMBL1907818)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50023980(2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-8-me...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024006((+)-2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50024006((+)-2-[(2,2-Dimethyl-cyclopropanecarbonyl)-amino]-...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against beta-lactamase renal dipeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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