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TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50408679(CHEMBL5287792)
Affinity DataKi:  0.00260nMAssay Description:Antagonist activity at cloned muscarinic M2 receptor-Gqi5 chimeric protein expressed in CHO cells assessed as acetylcholine-induced change in cytosol...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50408509(CHEMBL5277326)
Affinity DataKi:  0.00340nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50033531(CHEMBL333410 | N-[1-(2-Hydroxy-2-phenyl-ethyl)-3-m...)
Affinity DataKi:  0.00500nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM21865((14beta)-17-(cyclopropylmethyl)-18-(1-hydroxy-1-me...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50380909(CHEMBL2016678)
Affinity DataKi:  0.0490nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50102826(CHEMBL3339374)
Affinity DataKi:  0.0520nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50491882(CHEMBL3215908)
Affinity DataKi:  0.0520nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50033533(CHEMBL121403 | N-[(3R,4R)-1-((S)-2-Hydroxy-2-pheny...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM86416(Dmt-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  0.0636nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50491892(CHEMBL3216338)
Affinity DataKi:  0.0750nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50033534(CHEMBL338510 | N-[(3S,4S)-1-((S)-2-Hydroxy-2-pheny...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50491883(CHEMBL3216579)
Affinity DataKi:  0.0810nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50380906(CHEMBL2016675)
Affinity DataKi:  0.0970nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50177898(2-Fluoro-N-[4-methoxymethyl-1-(2-thiophen-2-yl-eth...)
Affinity DataKi:  0.100nMAssay Description:Binding constant for Opioid receptor mu 1 in mouseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50493749(CHEMBL2437063)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50395117(CHEMBL2163536)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned MOR-1 expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50491897(CHEMBL2387739)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50346951(CHEMBL1795711 | CHEMBL1795714)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned MOR-1 expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50493758(CHEMBL2437067)
Affinity DataKi:  0.120nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50189257(CHEMBL378753 | NalBzOH)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM21865((14beta)-17-(cyclopropylmethyl)-18-(1-hydroxy-1-me...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506207(CHEMBL4466064)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50491884(CHEMBL3216801)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50102828(CHEMBL3339372)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50033536(CHEMBL121494 | N-[(3R,4R)-1-((R)-2-Hydroxy-2-pheny...)
Affinity DataKi:  0.130nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50491885(CHEMBL2387740)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506210(CHEMBL4455793)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506217(CHEMBL4458688)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50102833(CHEMBL3339378)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506225(CHEMBL4562210)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.143nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM86416(Dmt-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  0.145nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50493755(CHEMBL2437064)
Affinity DataKi:  0.150nMAssay Description:Displacement of [125I]-BNtxA from mouse cloned mu opioid receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506211(CHEMBL4444746)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506219(CHEMBL4460495)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50102830(CHEMBL3339381)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50033530(CHEMBL121211 | N-[(3S,4S)-1-((R)-2-Hydroxy-2-pheny...)
Affinity DataKi:  0.150nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50033530(CHEMBL121211 | N-[(3S,4S)-1-((R)-2-Hydroxy-2-pheny...)
Affinity DataKi:  0.150nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.151nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50586108(CHEMBL5094608)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-naloxone from mouse mu opioid receptor expressed in CHO cell membranes assessed as inhibition constant incubated for 1.5 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506228(CHEMBL4570108)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506231(CHEMBL4575933)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.161nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.163nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50508336(CHEMBL4530500)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]-naloxone from mouse MOR expressed in CHO cell membranes by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506218(CHEMBL4565323)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50586084(CHEMBL5094575)
Affinity DataKi:  0.170nMAssay Description:Binding affinity to mouse mu opioid receptor expressed in CHO cells in presence of naltrexone incubated for 1.5 hrs by competitive radioligand bindin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM86418(Dmt-d-Ala-Phe-Phe-NH2)
Affinity DataKi:  0.173nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM86418(Dmt-d-Ala-Phe-Phe-NH2)
Affinity DataKi:  0.174nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50506213(CHEMBL4457013)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]-Naloxone from mouse mu opioid receptor expressed in CHO cells incubated for 1.5 hrs by competitive radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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