Compile Data Set for Download or QSAR
Report error Found 19 of ec50 for UniProtKB: Q9R0C9
LigandPNGBDBM50367061(NALORPHINE HYDROCHLORIDE | NALORPHINE)
Affinity DataEC50:  1.5nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataEC50:  3nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225937(CHEMBL3038189)
Affinity DataEC50:  6nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225933(CHEMBL2310921)
Affinity DataEC50:  6nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225936(CHEMBL3038190)
Affinity DataEC50:  7nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225935(CHEMBL2310915)
Affinity DataEC50:  7nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225940(CHEMBL2310917)
Affinity DataEC50:  50nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225942(CHEMBL2310916)
Affinity DataEC50:  90nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225932(CHEMBL2310918)
Affinity DataEC50:  90nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225934(CHEMBL2310922)
Affinity DataEC50:  100nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225938(CHEMBL2310919)
Affinity DataEC50:  100nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225939(CHEMBL3038192)
Affinity DataEC50:  130nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225941(CHEMBL2310920)
Affinity DataEC50:  130nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
LigandPNGBDBM50225931(CHEMBL3038191)
Affinity DataEC50:  180nMAssay Description:Displacement of [3H]dalamid ([D-Ala2,Met5] enkephalinamide) from opioid receptors of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2018
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50170660(CHEMBL521582 | [2-(4-Methoxy-3-phenethyloxy-phenyl...)
Affinity DataEC50:  1.07E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50179277(CHEMBL544343 | CHEMBL323056 | 1-(4-(6-methoxynapht...)
Affinity DataEC50:  1.50E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50179271(CHEMBL175560 | CHEMBL535366 | 1-(4-(6-methoxynapht...)
Affinity DataEC50:  1.94E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50179280(CHEMBL176941 | CHEMBL545278 | 1-(4-(6-methoxynapht...)
Affinity DataEC50:  2.55E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50179260(CHEMBL537177 | 1-(3-(6-methoxynaphthalen-1-yl)prop...)
Affinity DataEC50:  4.02E+4nMAssay Description:Antiproliferative activity mediated by sigma 1 receptor in rat C6 glioma cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed