Compile Data Set for Download or QSAR
Found 12 of ki for UniProtKB: Q09472
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50346552(CHEMBL1797936)
Affinity DataKi:  400nMAssay Description:Inhibition of synthetic VMA-tagged p300 (1287 to 1652 residues) (unknown origin) expressed in Escherichia coli BL21(RIL)-DE3 cells using H4-15 peptid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50346552(CHEMBL1797936)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of p300 HATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50456444(CHEMBL3734823)
Affinity DataKi:  400nMAssay Description:Inhibition of VMA intein chitin binding domain-fused p300 HAT domain (1287 to 1652 residues) (unknown origin) expressed in Escherichia coli BL21(RIL)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50346552(CHEMBL1797936)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of p300 HAT domain (unknown origin) using varying concentrations of acetyl-CoA and constant concentration of H4-15 as substrat...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50453820(CHEMBL4208500)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of VMA intein chitin binding domain-fused p300 HAT domain M1652G mutant (unknown origin) expressed in Escherichia coli BL21(RI...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50081125(CHEMBL3421961)
Affinity DataKi:  2.00E+3nMAssay Description:Noncompetitive inhibition of P300 (unknown origin) using acetyl CoA as substrate after 15 mins by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300/Hypoxia-inducible factor 1-alpha(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50537295(CHEMBL4524475)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of HIF-1alpha (786 to 826 residues) (unknown origin)/p300 (unknown origin) protein-protein interaction by ITCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50241990(CHEMBL502489 | Camboginol | Garcinol | Garcinol, 1)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50265449((1R,3S,9S,11R)-7-(3-Hydroxy-4-methoxy-benzoyl)-4,4...)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50081125(CHEMBL3421961)
Affinity DataKi:  9.40E+3nMAssay Description:Noncompetitive inhibition of P300 (unknown origin) using biotinylated H3 as substrate after 15 mins by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
University of Freiburg

Curated by ChEMBL
LigandPNGBDBM50260093(CHEMBL4078100)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human EP300 expressed in bacterial expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed