Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.158nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptor expressed in CHO-K1 cells after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Displacement of [3H]4-DAMP from human recombinant muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Displacement of [3H]4-DAMP from human recombinant M5 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Compound was evaluated for its binding affinity at human muscarinic receptor m5 by the displacement of [3H]-NMS radioligand using membranes from tran...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Evaluated for its binding affinity at human muscarinic receptor m5 by the displacement of [3H]NMS binding using membranes from transfected chinese ha...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Binding affinity to human M5 muscarinic receptor expressed in cell mebranes by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Antagonist activity at human muscarinic M5 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 109nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 119nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 134nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 143nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 148nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 149nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 159nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 168nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells in the presence of acetylcholine by calcium mobilisation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 194nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 215nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 222nMAssay Description:Displacement of [3H]NMS binding to human Muscarinic acetylcholine receptor M5 using membranes from transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 227nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair
Affinity DataIC50: 227nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization by Fl...More data for this Ligand-Target Pair