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Report error Found 430 of affinity data for UniProtKB/TrEMBL: P35869
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23936(1,3-dichloro-5-[(E)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to AhR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23940(1,3-dimethoxy-5-[(Z)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23941(1,3-dichloro-5-[(Z)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23940(1,3-dimethoxy-5-[(Z)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23946(1-[(Z)-2-(4-ethoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23947(1-[(Z)-2-(4-butoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23949(1,3-dichloro-5-[(Z)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23941(1,3-dichloro-5-[(Z)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23947(1-[(Z)-2-(4-butoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23949(1,3-dichloro-5-[(Z)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23946(1-[(Z)-2-(4-ethoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  12nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50605060(CHEMBL5198290 | US11891386, Compound 004)
Affinity DataKi:  88nMAssay Description:Binding affinity to AhR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50506041(CHEBI:16946 | L-kynurenine)
Affinity DataKi:  2.16E+4nMAssay Description:Inhibition of AhR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23945(1-[(Z)-2-(4-fluorophenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  1.04E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23940(1,3-dimethoxy-5-[(Z)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataKi:  1.33E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23946(1-[(Z)-2-(4-ethoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  1.54E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23943(1,3-difluoro-5-[(Z)-2-(4-fluorophenyl)ethenyl]benz...)
Affinity DataKi:  1.59E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23944(1,3-bis(trifluoromethyl)-5-[(Z)-2-[4-(trifluoromet...)
Affinity DataKi:  1.67E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23947(1-[(Z)-2-(4-butoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  2.33E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23951(1,3-dichloro-5-[(Z)-2-(3-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  4.17E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23942(1,3-difluoro-5-[(Z)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  4.55E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23935(1-[(E)-2-(4-butoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  5.01E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23950(1,3-dichloro-5-[(Z)-2-[3-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  5.27E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23948(1,3-dichloro-5-[(Z)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  7.14E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23941(1,3-dichloro-5-[(Z)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  7.69E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23949(1,3-dichloro-5-[(Z)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  8.34E+7nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23930(1,3-difluoro-5-[(E)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  1.09E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23928(1,3-dimethoxy-5-[(E)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataKi:  1.30E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23938(1,3-dichloro-5-[(E)-2-[3-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  1.47E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23939(1,3-dichloro-5-[(E)-2-(3-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  1.75E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23934(1-[(E)-2-(4-ethoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  2.00E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23936(1,3-dichloro-5-[(E)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  2.00E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23931(1,3-difluoro-5-[(E)-2-(4-fluorophenyl)ethenyl]benz...)
Affinity DataKi:  2.64E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23933(1-[(E)-2-(4-fluorophenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  3.23E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23932(1,3-bis(trifluoromethyl)-5-[(E)-2-[4-(trifluoromet...)
Affinity DataKi:  4.76E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23937(1,3-dichloro-5-[(E)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  7.14E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23929(1,3-dichloro-5-[(E)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  8.32E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM23929(1,3-dichloro-5-[(E)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  8.34E+8nMAssay Description:Binding affinity to aryl hydrocarbon receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50612694(CHEMBL5281742)
Affinity DataIC50:  0.885nMAssay Description:Antagonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50506040(CHEMBL4536502)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H] 3-MC from AhR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50240990(2-(3,4-dimethoxyphenyl)-5-fluorobenzothiazole | 5-...)
Affinity DataIC50:  25nMAssay Description:Binding affinity to AhR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)
Affinity DataIC50:  28nMAssay Description:Inhibition of aryl hydrocarbon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50525572(CH-223191 | CHEMBL1743245)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at AhR (unknown origin) assessed as inhibition of TCDD-induced luciferase activityMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50612692(CHEMBL5266911)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at AhR (unknown origin) expressed in human U87 cells assessed as inhibition of kynurenic acid-induced transactivation by Renilla/...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50612695(CHEMBL5271453)
Affinity DataIC50:  82nMAssay Description:Antagonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50612699(CHEMBL4303221)
Affinity DataIC50:  127nMAssay Description:Antagonist activity at AhR in human HepG2 cells assessed as inhibition of TCDD-induced receptor activation pretreated for 1 hr followed by TCDD addit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50612696(CHEMBL5280174)
Affinity DataIC50: <500nMAssay Description:Antagonist activity at AhR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50269353(CHEMBL4105559)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at human AhR expressed in Saccharomyces cerevisiae W303-1A (ATCC 208352) transformed with an episomal plasmid containing a minima...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50525572(CH-223191 | CHEMBL1743245)
Affinity DataIC50:  2.43E+3nMAssay Description:Antagonist activity at AhR in human HepG2 cells assessed as inhibition of FICZ-induced AhR transcriptional activity incubated for 24 hrs by Quanti-Lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAryl hydrocarbon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50191420((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-piperazin-1-yl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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