Compile Data Set for Download or QSAR
Report error Found 23 of ec50 for UniProtKB: Q6RI86
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50318486(CHEMBL422704 | 2-Methyl-2-(4-methyl-pent-3-enyl)-7...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50318487(Cannabigerol | CHEMBL497318)
Affinity DataEC50:  700nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633563(CHEMBL5421918)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50203072(Allylisothiocyanate | 3-isothiocyanatoprop-1-ene |...)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633568(CHEMBL5432734)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633564(CHEMBL5433171)
Affinity DataEC50:  6.90E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50541574(CHEMBL4636830)
Affinity DataEC50:  7.80E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50532217(CHEBI:67081 | Cannabigerolic Acid)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633562(CHEMBL5410813)
Affinity DataEC50:  8.50E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633567(CHEMBL5424611)
Affinity DataEC50:  8.80E+3nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633565(CHEMBL5437877)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622241(CHEMBL5416035)
Affinity DataEC50:  1.04E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622261(CHEMBL5432262)
Affinity DataEC50:  1.07E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622257(CHEMBL5412004)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633560(CHEMBL5415604)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633561(CHEMBL5404503)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622249(CHEMBL5428602)
Affinity DataEC50:  1.87E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622240(CHEMBL5416647)
Affinity DataEC50:  2.71E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622248(CHEMBL89848)
Affinity DataEC50:  2.72E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50633566(CHEMBL5404545)
Affinity DataEC50:  2.83E+4nMAssay Description:Agonist activity at rat TRPA1 transfected in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo4-AM dye based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622243(CHEMBL5417996)
Affinity DataEC50:  3.03E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622253(CHEMBL5410131)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50622247(CHEMBL5426686)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at rat recombinant TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed