Compile Data Set for Download or QSAR
maximum 50k data
Found 16 of ec50 for UniProtKB: A2AJP1
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataEC50:  27nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataEC50:  40nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50082042(CHEMBL139536 | N-(2,2,4,4-Tetramethyl-thiochroman-...)
Affinity DataEC50:  84nMAssay Description:Transcriptional activation of CV-1 cells expressing murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064253((2E,4Z,6Z)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50:  118nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataEC50:  200nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064255((2E,4Z,6Z)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50:  220nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50082041(4-iminomethylphenyl 4,4-dimethyl-6-chromanecarboxy...)
Affinity DataEC50:  294nMAssay Description:Transcriptional activation of CV-1 cells expressing murine Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50293410((E)-3-[5'-(Adamant-1-yl)-2-chloro-4'-hydroxy-2'-me...)
Affinity DataEC50:  576nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50293413((E)-3-[5'-(Adamant-1-yl)-2-chloro-4'-[(2-methoxyet...)
Affinity DataEC50:  600nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50293412(6-[5-(Adamant-1-yl)-4-[(2-methoxyethoxy)methoxy]-2...)
Affinity DataEC50:  667nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50293411(2-[5'-(Adamant-1-yl)-2-chloro-4'-[(2-methoxyethoxy...)
Affinity DataEC50:  1.14E+3nMAssay Description:Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064250((2E,4E,6E)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064252((2Z,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50064251((2Z,4E,6E)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Mus musculus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed