TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 352nMAssay Description:Positive modulation of Kca 1.1 (unknown origin)More data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 3.34E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 3.86E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 4.43E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 5.07E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 5.13E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 5.86E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 6.75E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 6.94E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 8.12E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 1.34E+4nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 1.51E+4nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Maxi-K channel (unknown origin) by thallium flux assayMore data for this Ligand-Target Pair