Compile Data Set for Download or QSAR
Report error Found 199 of ic50 for UniProtKB: Q9WUD2
LigandPNGBDBM50222640(CHEMBL415543)
Affinity DataIC50: 0.320nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222640(CHEMBL415543)
Affinity DataIC50: 0.320nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222695(CHEMBL155433)
Affinity DataIC50: 0.460nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222637(CHEMBL154743)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222696(CHEMBL156041)
Affinity DataIC50: 0.550nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222635(CHEMBL267205)
Affinity DataIC50: 0.720nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222647(CHEMBL154990)
Affinity DataIC50: 0.950nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222649(CHEMBL155730)
Affinity DataIC50: 0.950nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222641(CHEMBL157962)
Affinity DataIC50: 1.20nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222638(CHEMBL422702)
Affinity DataIC50: 2.40nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222644(CHEMBL434295)
Affinity DataIC50: 2.5nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222648(CHEMBL156693)
Affinity DataIC50: 3nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222639(CHEMBL356682)
Affinity DataIC50: 3.20nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222646(CHEMBL157917)
Affinity DataIC50: 5.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222694(CHEMBL158189)
Affinity DataIC50: 6.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222691(CHEMBL156927)
Affinity DataIC50: 9.30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222690(CHEMBL345157)
Affinity DataIC50: 10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222645(CHEMBL157918)
Affinity DataIC50: 11nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222693(CHEMBL157579)
Affinity DataIC50: 12nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50224228(CHEMBL46233)
Affinity DataIC50: 15nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224175(CHEMBL48061)
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50222634(CHEMBL157473)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222643(CHEMBL157688)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50222692(CHEMBL348634)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2018
Entry Details Article
PubMed
LigandPNGBDBM50224176(CHEMBL296963)
Affinity DataIC50: 30nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM20321(JYL1421 | CHEMBL388824 | 3-[(4-tert-butylphenyl)me...)
Affinity DataIC50: 37nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
LigandPNGBDBM20321(JYL1421 | CHEMBL388824 | 3-[(4-tert-butylphenyl)me...)
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224229(CHEMBL48998)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224232(CHEMBL296729)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224234(CHEMBL45252)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224196(CHEMBL43723)
Affinity DataIC50: 66nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224230(CHEMBL47282)
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224237(CHEMBL431341)
Affinity DataIC50: 70nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMed
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM20315(3-[(4-tert-butylphenyl)methyl]-1-[(4-methanesulfon...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463972(CHEMBL4249976)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50224239(CHEMBL295773)
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM20460(N-Vannilyloleoylamide | (Z)-N-[(4-hydroxy-3-methox...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50224100(CHEMBL44057)
Affinity DataIC50: 220nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224235(CHEMBL45417)
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463948(CHEMBL4249973)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50223778(CHEMBL164875)
Affinity DataIC50: 300nMAssay Description:In vitro antagonist activity at the vanilloid receptor in rat DRG neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2018
Entry Details Article
PubMed
LigandPNGBDBM50224226(CHEMBL45455)
Affinity DataIC50: 320nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224238(CHEMBL47602)
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463944(CHEMBL1672687)
Affinity DataIC50: 490nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50224195(CHEMBL48102)
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50224194(CHEMBL47473)
Affinity DataIC50: 580nMAssay Description:In vitro inhibitory concentration was determined against [45Ca2+]- influx in rat DRG neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details Article
PubMed
LigandPNGBDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataIC50: 590nMAssay Description:Inhibition of [Ca2+] uptake in dorsal root ganglion (DRG) neurons from neonatal Sprague-Dawley ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM20284(N-[2-(4-chlorophenyl)ethyl]-7,8-dihydroxy-2,3,4,5-...)
Affinity DataIC50: 600nMAssay Description:Ability to inhibit [Ca2+] influx neonatal rat cultured spinal sensory neurons.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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