Compile Data Set for Download or QSAR
Report error Found 236 of ic50 for UniProtKB: Q02485
LigandPNGBDBM50029417([4-(4-Methoxy-phenyl)-4H-benzo[b]pyrrolo[1,2-d][1,...)
Affinity DataIC50: 0.420nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details

LigandPNGBDBM50306490((+)-(S)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50: 0.420nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50: 0.760nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50469633(CHEMBL21906)
Affinity DataIC50: 0.780nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptors (CCRs) from rat cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2020
Entry Details Article

LigandPNGBDBM50103634(CL-287389 | FK-235 | Nilvadipine | Nivadipine | SK...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Voltage-dependent L-type calcium channel in rat thoracic aorta ringMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
LigandPNGBDBM50306490((+)-(S)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50: 1.48nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50229256(CHEMBL73590)
Affinity DataIC50: 1.60nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50227967(CHEMBL78973)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [3H]- Nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 2.57nMAssay Description:Inhibition of L-type calcium channel in Rattus norvegicus Wistar (rat) thoracic aorta assessed as relaxation of KCl-induced vasoconstriction after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of L-type calcium channel in Rattus norvegicus Wistar (rat) thoracic aorta assessed as relaxation of KCl-induced vasoconstriction after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50101815(CHEBI:7550 | Nicardipine)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50475660(CHEMBL201566)
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50: 3.62nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50475658(CHEMBL201984)
Affinity DataIC50: 3.70nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475653(CHEMBL382528)
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475650(CHEMBL203041)
Affinity DataIC50: 6.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50479255(CHEMBL453084)
Affinity DataIC50: 7nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
LigandPNGBDBM50227968(CHEMBL310953)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of [3H]- Nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50: 8.14nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cardiac membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50227969(CV-4093 | CHEMBL312176)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of [3H]- Nitrendipine binding to L-type calcium channels of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50475663(CHEMBL202464)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475664(CHEMBL369934)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50229315(CHEMBL312304)
Affinity DataIC50: 10nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50475672(CHEMBL201057)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475662(CHEMBL201860)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50280077(sec-Butyl-[4-(2,4-dimethoxy-phenyl)-4H-benzo[b]pyr...)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details

LigandPNGBDBM50306489((-)-(R)-3-methyl 5-pentyl 2,6-dimethyl-4-(3-nitrop...)
Affinity DataIC50: 17.6nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor in rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50475669(CHEMBL382072)
Affinity DataIC50: 20nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
LigandPNGBDBM50475669(CHEMBL382072)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475656(CHEMBL201306)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50227617(CHEMBL46635)
Affinity DataIC50: 20nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50229269(CHEMBL72696)
Affinity DataIC50: 21nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50229269(CHEMBL72696)
Affinity DataIC50: 21nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50227621(CHEMBL46452)
Affinity DataIC50: 26nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50229288(CHEMBL75494)
Affinity DataIC50: 27nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50227619(CHEMBL44275)
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 28nMAssay Description:Inhibition of L-type calcium channel in Rattus norvegicus Wistar (rat) thoracic aorta assessed as relaxation of phenylephrine-induced vasoconstrictio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 28nMAssay Description:Inhibition of L-type calcium channel in Rattus norvegicus Wistar (rat) thoracic aorta assessed as relaxation of phenylephrine-induced vasoconstrictio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PDB3D3D Structure (crystal)
LigandPNGBDBM50475661(CHEMBL204486)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50227627(CHEMBL295323)
Affinity DataIC50: 31nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227615(CHEMBL46590)
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50229332(CHEMBL72341)
Affinity DataIC50: 33nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50229310(CHEMBL73583)
Affinity DataIC50: 36nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50229270(CHEMBL306566)
Affinity DataIC50: 37nMAssay Description:Affinity to bind dihydropyridine receptor (DHP receptor) by inhibiting the radioligand [3H]nitrendipineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2019
Entry Details Article
PubMed
LigandPNGBDBM50004704(Acetic acid 5-(2-dimethylamino-ethyl)-2-(4-methoxy...)
Affinity DataIC50: 42nMAssay Description:Displacement of [3H]nitrendipine from calcium channel receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2018
Entry Details
PDB3D3D Structure (crystal)
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