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TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50539801(CHEMBL4648912 | US11840533, Compound 70)
Affinity DataKd: <1nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  12nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataKd:  14nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512964(CHEMBL4574669)
Affinity DataKd:  78nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512976(CHEMBL4543497)
Affinity DataKd:  85nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512965(CHEMBL4453637)
Affinity DataKd:  100nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512979(CHEMBL4457684)
Affinity DataKd:  103nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512968(CHEMBL4454700)
Affinity DataKd:  106nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512967(CHEMBL4449143)
Affinity DataKd:  118nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512966(CHEMBL4570924)
Affinity DataKd:  120nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512980(CHEMBL4570969)
Affinity DataKd:  126nMAssay Description:Binding affinity to human PCAF bromodomain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512960(CHEMBL4545594)
Affinity DataKd:  128nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512954(CHEMBL4527339)
Affinity DataKd:  138nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512958(CHEMBL4439202)
Affinity DataKd:  140nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512975(CHEMBL4471748)
Affinity DataKd:  152nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512959(CHEMBL4454766)
Affinity DataKd:  183nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512962(CHEMBL4565832)
Affinity DataKd:  215nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512969(CHEMBL4539318)
Affinity DataKd:  233nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512961(CHEMBL4541223)
Affinity DataKd:  242nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataKd:  300nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50584925(CHEMBL5079885)
Affinity DataKd: <316nMAssay Description:Binding affinity to human PCAF bromodomain assessed as dissociation constant by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512978(CHEMBL4544739)
Affinity DataKd:  347nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataKd:  370nMAssay Description:Binding affinity to PCAF (unknown origin) by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512987(CHEMBL4525423)
Affinity DataKd:  535nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512972(CHEMBL4579627)
Affinity DataKd:  621nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512977(CHEMBL4453013)
Affinity DataKd:  676nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512970(CHEMBL4470046)
Affinity DataKd:  820nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512984(CHEMBL4547880)
Affinity DataKd:  935nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human PCAF (G715 to D831 residues) expressed in mammalian expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2019
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512973(CHEMBL4438712)
Affinity DataKd:  1.19E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512982(CHEMBL4528565)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512988(CHEMBL4556786)
Affinity DataKd:  2.16E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512981(CHEMBL4449886)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512956(CHEMBL4437954)
Affinity DataKd:  3.04E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512983(CHEMBL4537244)
Affinity DataKd:  3.41E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM179481(US9675697, Cpd. No. 73)
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50504160(CHEMBL3133807 | US11773085, Compound B25)
Affinity DataKd:  4.76E+3nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: G715-D831More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOScan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50150068(CHEMBL3775323)
Affinity DataKd:  6.80E+3nMAssay Description:Displacement of biotinylated small molecule ligand from His/FLAG-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) after 15 mins by Alph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50150068(CHEMBL3775323)
Affinity DataKd:  6.80E+3nMAssay Description:Binding affinity to N-terminal His-tagged PCAF (715 to 831 residues) (unknown origin) expressed in Escherichia coli Rosetta cells by isothermal titra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512955(CHEMBL4454395)
Affinity DataKd:  7.80E+3nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512985(CHEMBL4584442)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512986(CHEMBL4581184)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50615275(CHEMBL5282240)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM321437((E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50615276(CHEMBL5270178)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM321424(6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512971(CHEMBL4471746)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512974(CHEMBL4471600)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512957(CHEMBL4460616)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
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