Compile Data Set for Download or QSAR
Found 92 of ic50 for UniProtKB: P41586
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50550811(CHEMBL4740931)
Affinity DataIC50: <0.0100nMAssay Description:Antagonist activity at PAC1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced inhibition of CREB phosphorylati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50596676(CHEMBL5203375)
Affinity DataIC50:  0.110nMAssay Description:Antagonist activity at PAC-1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced increase in intracellular cAMP ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50550810(CHEMBL4757203)
Affinity DataIC50:  0.182nMAssay Description:Antagonist activity at PAC1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced inhibition of CREB phosphorylati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50596675(CHEMBL5208587)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity at PAC-1 receptor (unknown origin) expressed in CHO cells assessed as inhibition of PACAP-induced increase in intracellular cAMP ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50200209(CHEMBL219499)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]PACAP27 from human PAC1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50606528(CHEMBL5219662)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at PAC1R in human SH-SY5Y cells assessed as inhibition of PACAP38-induced cAMP accumulation pre-incubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250033(CHEMBL525419 | [Ala7]PACAP38)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250074(CHEMBL507480 | [Bip6]PACAP27)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250018(CHEMBL524852 | PACAP27)
Affinity DataIC50:  4.60nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human PAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250034(CHEMBL499781 | [D-His1]PACAP27)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250077(CHEMBL503123 | [Nal6]PACAP38)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250022(CHEMBL525392 | [Ala2]PACAP27)
Affinity DataIC50:  5.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250035(CHEMBL525073 | [D-His1]PACAP38)
Affinity DataIC50:  5.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250075(CHEMBL526315 | [Bip6]PACAP38)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250059(Ac-PACAP38 | CHEMBL530563)
Affinity DataIC50:  5.70nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250019(CHEMBL524658 | PACAP | PACAP(1-38) | PACAP-38 | PA...)
Affinity DataIC50:  6.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250076(CHEMBL525613 | [Nal6]PACAP27)
Affinity DataIC50:  6.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250037(CHEMBL524894 | [D-Ser2]PACAP38)
Affinity DataIC50:  6.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250071(CHEMBL524683 | [Cha6]PACAP38)
Affinity DataIC50:  6.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250073(CHEMBL526360 | [Tyr6]PACAP38)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250069(CHEMBL524494 | [Glu3]PACAP38)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250085(CHEMBL506517 | [Aib2]PACAP38)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250039(CHEMBL524334 | [D-Asp3]PACAP38)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250036(CHEMBL506133 | [D-Ser2]PACAP27)
Affinity DataIC50:  7.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250061(CHEMBL498948 | [His(1-Me)1]PACAP38)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250078(CHEMBL524672 | [Pro2]PACAP27)
Affinity DataIC50:  7.80nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250072(CHEMBL498867 | [Tyr6]PACAP27)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250023(CHEMBL500280 | [Ala2]PACAP(1-38) | [Ala2]PACAP38)
Affinity DataIC50:  7.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250058(Ac-PACAP27 | CHEMBL505046)
Affinity DataIC50:  8.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250018(CHEMBL524852 | PACAP27)
Affinity DataIC50:  8.30nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250079(CHEMBL506840 | [Pro2]PACAP38)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250080(CHEMBL524495 | [Hyp2]PACAP27)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250081(CHEMBL499507 | [Hyp2]PACAP38)
Affinity DataIC50:  8.60nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250026(CHEMBL526899 | [Ala4]PACAP27)
Affinity DataIC50:  9.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250047(CHEMBL525591 | [N-Me-Ser2]PACAP38)
Affinity DataIC50:  9.10nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250087(CHEMBL499665 | [Aib4]PACAP38)
Affinity DataIC50:  9.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250065(CHEMBL502352 | [Asn3]PACAP38)
Affinity DataIC50:  9.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250046(CHEMBL525258 | [N-Me-Ser2]PACAP27)
Affinity DataIC50:  9.40nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250084(CHEMBL500227 | [Aib2]PACAP27)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250027(CHEMBL525091 | [Ala4]PACAP38)
Affinity DataIC50:  9.84nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250038(CHEMBL509368 | [D-Asp3]PACAP27)
Affinity DataIC50:  9.90nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250049(CHEMBL502619 | [N-Me-Asp3]PACAP38)
Affinity DataIC50:  10.4nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250068(CHEMBL501240 | PACAP(1-27) | PACAP-27 | [Glu3]PACA...)
Affinity DataIC50:  10.6nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250032(CHEMBL445530 | [Ala7]PACAP27)
Affinity DataIC50:  10.8nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250070(CHEMBL524471 | [Cha6]PACAP27)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250063(CHEMBL508607 | [His(3-Me)1]PACAP38)
Affinity DataIC50:  11.3nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250067(CHEMBL526000 | [Aad3]PACAP38)
Affinity DataIC50:  12.5nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250060(CHEMBL526131 | [His(1-Me)1]PACAP27)
Affinity DataIC50:  15.6nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250062(CHEMBL524675 | [His(3-Me)1]PACAP27)
Affinity DataIC50:  21.6nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
University of Toyama

Curated by ChEMBL
LigandPNGBDBM50250048(CHEMBL525207 | [N-Me-Asp3]PACAP27)
Affinity DataIC50:  25.2nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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