Compile Data Set for Download or QSAR
Report error Found 950 of ki for UniProtKB: P07550
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595424(CHEMBL5172865)
Affinity DataKi:  0.00398nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50379086(CHEMBL2012522 | CHEMBL2012521 | LY-377604)
Affinity DataKi:  0.0120nMAssay Description:Displacement of [125I]Iodocyanopindolol from human adrenergic beta2 receptor expressed in insect sf9 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569290(CHEMBL4871517)
Affinity DataKi:  0.0126nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569294(CHEMBL4863525)
Affinity DataKi:  0.0158nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595404(CHEMBL5184455)
Affinity DataKi:  0.0200nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595423(CHEMBL5190387)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595426(CHEMBL5193853)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595427(CHEMBL5200887)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569293(CHEMBL4874819)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50167072(CHEMBL3799125)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50027663(Carazolol | 1-(9H-carbazol-4-yloxy)-3-(isopropylam...)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50167072(CHEMBL3799125)
Affinity DataKi:  0.0340nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569292(CHEMBL4857743)
Affinity DataKi:  0.0398nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595403(CHEMBL5208201)
Affinity DataKi:  0.0398nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to human beta 2 adrenergic receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595405(CHEMBL5184598)
Affinity DataKi:  0.0501nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595425(CHEMBL5208957)
Affinity DataKi:  0.0501nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569299(CHEMBL4866806)
Affinity DataKi:  0.0501nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50526679(CHEMBL4456301)
Affinity DataKi:  0.0730nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM85818(Fluorocarazolol,(S) | Fluorocarazolol,(R))
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569300(CHEMBL4871702)
Affinity DataKi:  0.100nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569295(CHEMBL4854418)
Affinity DataKi:  0.100nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50098668(4-(3-tert-Butylamino-2-hydroxy-propoxy)-1,3-dihydr...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 2 adrenergic receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50318987(1-(9H-carbazol-4-yloxy)-3-(4-(pyridin-3-ylmethyl)p...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50027663(Carazolol | 1-(9H-carbazol-4-yloxy)-3-(isopropylam...)
Affinity DataKi:  0.114nMAssay Description:Displacement of [3H]DHA from human beta2 adrenoceptor by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM85818(Fluorocarazolol,(S) | Fluorocarazolol,(R))
Affinity DataKi:  0.138nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50274012(1-tert-Butylamino-3-(dibenzofuran-1-yloxy)-propan-...)
Affinity DataKi:  0.145nMAssay Description:Displacement of [3H]DHA from human beta2 adrenoceptor by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569302(CHEMBL4878138)
Affinity DataKi:  0.158nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50526681(CHEMBL4537221)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM25759([3-(9H-carbazol-4-yloxy)-2-hydroxypropyl][2-(2-met...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity to human beta 2 adrenergic receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569297(CHEMBL4846536)
Affinity DataKi:  0.200nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569296(CHEMBL4852629)
Affinity DataKi:  0.200nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50318988((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50318986(1-(9H-carbazol-4-yloxy)-3-(4-(4-methoxybenzyl)pipe...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50318989((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50292219((2S)-1-(tert-butylamino)-3-[(4-morpholin-4-yl-1,2,...)
Affinity DataKi:  0.209nMAssay Description:Displacement of [3H]-CGP12177 from human beta2 ADR expressed in HEK293T cell membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50166979(CHEMBL3798748)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569301(CHEMBL4854091)
Affinity DataKi:  0.251nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569298(CHEMBL4878395)
Affinity DataKi:  0.251nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50569301(CHEMBL4854091)
Affinity DataKi:  0.251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50318990((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperi...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50324835((R)-4-hydroxy-7-(1-hydroxy-2-(3-(methyl(phenyl)ami...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50274013(1-(4-benzhydrylpiperazin-1-yl)-3-(3-methyl-1H-indo...)
Affinity DataKi:  0.300nMAssay Description:Displacement of radioligand from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)
Affinity DataKi:  0.302nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50274013(1-(4-benzhydrylpiperazin-1-yl)-3-(3-methyl-1H-indo...)
Affinity DataKi:  0.311nMAssay Description:Displacement of [3H]DHA from human beta2 adrenoceptor by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50019443(LB-46 | 1-(1H-Indol-4-yloxy)-3-isopropylamino-prop...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity to human beta 2 adrenergic receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
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