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TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.00800nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86812(NSC_45263784 | CAS_45263784 | rac-2-(6-fluoro-5-(4...)
Affinity DataKi:  0.00900nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049750(CHEMBL59986 | (S)-3-(azetidin-2-ylmethoxy)pyridine...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50066789(A-85380,5-Iodo | CHEMBL123433 | A-85380-I | 3-((S)...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50263171((+)-2-(6'-[18F]fluoro-3,3'-bipyridin-5-yl)-7-methy...)
Affinity DataKi:  0.0110nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50216315((1R,4R)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[...)
Affinity DataKi:  0.0180nMAssay Description:Displacement of [3H]cytosine form alpha4beta2 nAChR in rat striatumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50263095((+/-)-7-Methyl-2-exo-[3'-(2-fluoropyridin-4-yl)-5'...)
Affinity DataKi:  0.0190nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50100712(IPH | Epibatidine-I,(+/-) | CHEMBL54586 | 2-(6-Iod...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50100717(2-(pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane | CHE...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50275878(3-(6-chloropyridin-3-yl)-3,6-diazabicyclo[3.1.1]he...)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0260nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50295955(5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyrid...)
Affinity DataKi:  0.0280nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50295959((S)-2-chloro-5-((1-methylpyrrolidin-2-yl)methoxy)-...)
Affinity DataKi:  0.0280nMAssay Description:Displacement of [125I]5-A-85380 from alpha4beta2 nicotinic receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86815(CAS_45266019 | NSC_45266019 | rac-2-(6-fluoro-5-(4...)
Affinity DataKi:  0.0290nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50062639(CHEMBL439766 | ABT-594 | A-98593 | 5-((S)-1-Azetid...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0350nMAssay Description:Displacement of [3H]nicotine from alpha4beta2 nAChR in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50279404(cis-2-(5-Ethoxy-3-pyridinyl)octahydropyrrolo[3,4-c...)
Affinity DataKi:  0.0350nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50275880(3-(6-bromopyridin-3-yl)-3,6-diazabicyclo[3.1.1]hep...)
Affinity DataKi:  0.0390nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50279405(cis-3-(5-Propyloxy-3-pyridinyl)-3,7-diazabicyclo[3...)
Affinity DataKi:  0.0410nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86816(NSC_45263769 | CAS_45263769 | rac-2-(5-(4-chloroph...)
Affinity DataKi:  0.0440nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0460nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0470nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0470nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50062641(CHEMBL430497 | 5-((R)-1-Azetidin-2-ylmethoxy)-2-ch...)
Affinity DataKi:  0.0480nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50278878(cis-3-(5-Isopropyloxy-3-pyridinyl)-3,7-diazabicycl...)
Affinity DataKi:  0.0510nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86810(CAS_45266065 | NSC_45266065 | rac-2-(6-fluoro-5-(3...)
Affinity DataKi:  0.0530nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50295956(2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-m...)
Affinity DataKi:  0.0550nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50275879(3-(pyridin-3-yl)-3,6-diazabicyclo[3.1.1]heptane | ...)
Affinity DataKi:  0.0560nMAssay Description:Displacement of [3H]epibatidine form alpha4beta2 nAChR in rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50278877(cis-2-(5-(Benzyloxy)pyridin-3-yl)octahydropyrrolo[...)
Affinity DataKi:  0.0580nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50263130((+/-)-7-Methyl-2-exo-[3'-(2-fluoropyridin-3-yl)-5'...)
Affinity DataKi:  0.0580nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50066789(A-85380,5-Iodo | CHEMBL123433 | A-85380-I | 3-((S)...)
Affinity DataKi:  0.0590nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50279402(cis-2-(5-Bromopyridin-3-yl)-octahydro-pyrrolo[3,4-...)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0610nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0610nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0610nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50295954(2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-m...)
Affinity DataKi:  0.0620nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50295958((S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl...)
Affinity DataKi:  0.0620nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0720nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86805(CAS_45263788 | NSC_45263788 | rac-2-(5-(3-chloroph...)
Affinity DataKi:  0.0730nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50279403(cis-2-(5-Methoxy-3-pyridinyl)octahydropyrrolo[3,4-...)
Affinity DataKi:  0.0810nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86819(NSC_45263772 | CAS_45263772 | rac-2-(6-fluoro-5-(3...)
Affinity DataKi:  0.0870nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86817(CAS_45263779 | NSC_45263779 | rac-4-(5-(7-aza-bicy...)
Affinity DataKi:  0.0950nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86807(CAS_45263775 | NSC_45263775 | rac-3-(5-(7-aza-bicy...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM86818(CAS_45266054 | NSC_45266054 | rac-2-(6-fluoro-5-(3...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50166908(CHEMBL556954 | VARENICLINE | 5,8,14-triazatetracyc...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50279369(cis-2-(3-Pyridinyl)octahydropyrrolo[3,4-c]pyrrole ...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain minus cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50295953(2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50171347(A-85380 | CHEMBL190589 | 3-(Azetidin-2-ylmethoxy)-...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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