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Found 742 of ic50 for UniProtKB: P00749
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50147093(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataIC50:  0.620nMAssay Description:Inhibition of uPA (unknown origin)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194745(CHEMBL385900 | diphenyl 1-[(N-2-thiophenesulfonyl-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194741(CHEMBL385158 | diphenyl 1-[(N-benzenesulfonyl-D-se...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50:  3.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228418(CHEMBL393591 | methyl 1-(diphenoxyphosphoryl)-2-(4...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228412(CHEMBL393979 | methyl 1-(bis(4-acetamidophenoxy)ph...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228425(CHEMBL239118 | di-(4-acetamidophenyl) 1-(methylsul...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194743(CHEMBL214814 | diphenyl 1-[(N-alpha-toluenesulfony...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228420(CHEMBL391968 | di-(4-acetamidophenyl) 1-(benzyloxy...)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50145689(CHEMBL80844 | [1-[(S)-2-((R)-2-Benzyloxycarbonylam...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194737(CHEMBL384263 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194742(CHEMBL263977 | diphenyl 1-[(N-benzyl-D-seryl)-L-al...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194746(CHEMBL405546 | diphenyl 1-[(N-o-methylbenzoyl-D-se...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088978(CHEMBL176515 | N-[1-(1-Carbamimidoyl-2-hydroxy-pip...)
Affinity DataIC50:  5.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194734(CHEMBL386275 | diphenyl 1-[(N-p-methoxybenzenesulf...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194744(CHEMBL385897 | diphenyl 1-[(N-naphthalenesulfonyl-...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194736(CHEMBL189823 | diphenyl 1-[(N-o,o-dimethylbenzoyl-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194735(CHEMBL215961 | diphenyl 1-[(N-p-cyanobenzenesulfon...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194738(CHEMBL386249 | diphenyl 1-[(N-p-bromobenzenesulfon...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228421(CHEMBL238493 | diphenyl 1-(methylsulfonylamino)-2-...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50:  6.60nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194732(CHEMBL214539 | di-(4-acetamidophenyl) 1-[(N-benzyl...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of [3H]-FPP incorporation into biotin-linked K-ras decapeptide (CVIM) by bovine farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194739(CHEMBL213216 | diphenyl 1-[(N-2-thienyl-D-seryl)-L...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194740(CHEMBL404226 | diphenyl 1-[(N-p-methylbenzoyl-D-se...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228410(CHEMBL239535 | diphenyl 1-(benzyloxycarbonylamino)...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228414(CHEMBL239747 | diphenyl 1-acetamido-2-(4-guanidino...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228417(CHEMBL238491 | diphenyl 1-(o-toluenesulfonylamino)...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228423(CHEMBL239536 | ethyl 1-(diphenoxyphosphoryl)-2-(4-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50194733(CHEMBL411215 | diphenyl 1-[(N-1-adamantanyl-D-sery...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50:  10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50:  10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088979(CHEMBL366666 | {(R)-2-[2-((S)-1-Carbamimidoyl-2-hy...)
Affinity DataIC50:  11nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088985(CHEMBL369042 | {2-[2-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  12nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50:  14nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50301972(2-(6-(5-amino-3'-(aminomethyl)biphenyl-3-yloxy)-4-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50542728(CHEMBL4635912)
Affinity DataIC50:  16nMAssay Description:Inhibition of human urokinase using fluorescent peptide as substrate by florescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088977(CHEMBL177557 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  19nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50542731(CHEMBL4642845)
Affinity DataIC50:  20nMAssay Description:Inhibition of human uPA using fluorescent peptide as substrate by florescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50542732(CHEMBL4647925)
Affinity DataIC50:  20nMAssay Description:Inhibition of human uPA using fluorescent peptide as substrate by florescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50231520((R)-N-[(S)-1-(4-carbamimidoyl-benzylcarbamoyl)-2-h...)
Affinity DataIC50:  20nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50:  20nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50467209(CHEMBL4291446)
Affinity DataIC50:  23nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50088987(CHEMBL174813 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  23nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50301973(2-(6-(3'-(aminomethyl)-5-hydroxybiphenyl-3-yloxy)-...)
Affinity DataIC50:  23nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50301982(2-(6-(3'-(aminomethyl)biphenyl-3-yloxy)-4-(3-(dime...)
Affinity DataIC50:  25nMAssay Description:Inhibition of uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50184648(CHEMBL378976 | [benzyloxycarbonylamino-(4-guanidin...)
Affinity DataIC50:  26nMAssay Description:Inhibition of human uPA by chromogenic assay using Cbz-Val-Gly-Arg-pNA as chromogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50228426(CHEMBL391344 | diphenyl 1-(naphthalenesulfonylamin...)
Affinity DataIC50:  26.5nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1/Urokinase-type plasminogen activator(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM264615(US9718760, C182)
Affinity DataIC50:  33nMpH: 7.4 T: 2°CAssay Description:To determine the efficacy of various synthesized compounds as PAI-1 inhibitors, a fluorometric plate assay was carried out to measure the half maxima...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Wollongong

Curated by ChEMBL
LigandPNGBDBM50467207(CHEMBL4288828)
Affinity DataIC50:  34nMAssay Description:Inhibition of human uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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