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Report error Found 281 of ec50 for UniProtKB: O43613
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50586152(CHEMBL5079059)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at human OX1R expressed in CHO-K1 cells by FLIPR calcium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50439587(CHEMBL2418879)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at OX1 receptor (unknown origin) expressed in RD-HGA16 cells assessed as calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50439587(CHEMBL2418879)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at human OX1 receptor overexpressed in CHO-RD-HGA16 cells assessed as calcium mobilization after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121795(CHEMBL436915 | [Gly17]orexin-B)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121792(CHEMBL439541 | [D-Ala19]orexin-B)
Affinity DataEC50:  0.520nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121773(CHEMBL386549 | [D-Asn20]orexin-B)
Affinity DataEC50:  0.610nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121769(CHEMBL428123 | [D-Gln12]orexin-B)
Affinity DataEC50:  0.770nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121770(CHEMBL413504 | [Ala14]orexin-B)
Affinity DataEC50:  0.820nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121783(CHEMBL413434 | Orexin-B)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121809(CHEMBL410899 | [D-Pro5]orexin-B)
Affinity DataEC50:  0.850nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121791(CHEMBL410947 | [D-Pro4]orexin-B)
Affinity DataEC50:  0.890nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121806(CHEMBL265907 | [Ala9]orexin-B)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121777(CHEMBL265746 | [D-Ser2]orexin-B)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121794(CHEMBL427771 | [Ala7]orexin-B)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121778(CHEMBL265423 | [D-Ala3]orexin-B)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121793(CHEMBL264342 | [D-Ala6]orexin-B)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121775(CHEMBL438036 | [D-Leu7]orexin-B)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121810(CHEMBL409301 | [D-Ala9]orexin-B)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121796(CHEMBL414312 | [Ala16]orexin-B)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121815(CHEMBL410480 | [Ala6]orexin-B)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121766(CHEMBL410816 | [D-Arg1]orexin-B)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121765(CHEMBL437464 | [Ala13]orexin-B)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121803(CHEMBL265404 | [Ala3]orexin-B)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121790(CHEMBL409456 | [Ala1]orexin-B)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121780(CHEMBL414332 | [Ala2]orexin-B)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121767(CHEMBL409970 | [D-Ala17]orexin-B)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121761(CHEMBL441008 | [Ala8]orexin-B)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121759(CHEMBL438587 | [D-Leu15]orexin-B)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121786(CHEMBL442505 | [Ala5]orexin-B)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121797(CHEMBL437274 | [Ala4]orexin-B)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121784(CHEMBL266409 | [Ala12]orexin-B)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121785(CHEMBL411174 | [D-Arg13]orexin-B)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121772(CHEMBL413284 | [D-Gln8]orexin-B)
Affinity DataEC50:  4nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121817(CHEMBL437149 | [Trp11]orexin-B)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121798(CHEMBL413884 | [Ala21]orexin-B)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121760(CHEMBL413285 | [D-Gln16]orexin-B)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121811(CHEMBL440060 | [Ala18]orexin-B)
Affinity DataEC50:  6nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121774(CHEMBL264343 | [D-Leu11]orexin-B)
Affinity DataEC50:  7nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121776(CHEMBL430313 | [D-His21]orexin-B)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121781(CHEMBL275985 | [Gly22]orexin-B)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121764(CHEMBL411116 | [D-Ser18]orexin-B)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121788(CHEMBL441918 | [Ala11]orexin-B)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50445183(CHEMBL438397)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at human OX1 receptor overexpressed in CHO-RD-HGA16 cells assessed as calcium mobilization after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121805(CHEMBL430064 | [Ala10]orexin-B)
Affinity DataEC50:  9.10nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121763(CHEMBL410960 | [D-Arg10]orexin-B)
Affinity DataEC50:  9.80nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121808(CHEMBL263628 | [Ala19]orexin-B)
Affinity DataEC50:  14nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50596486(CHEMBL5203887)
Affinity DataEC50:  14nMAssay Description:Agonist activity at OX1R (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121799(CHEMBL409967 | [Gly23]orexin-B)
Affinity DataEC50:  22nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50121802(CHEMBL439288 | [D-Ala22]orexin-B)
Affinity DataEC50:  22nMAssay Description:Agonist activity against human orexin 1 receptor; EC50; nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50579705(CHEMBL5070320)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human OX1R stably expressed in CHO RD-HGA16 cells assessed as fluorescence changes measured after 30 mins by calcium mobilization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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