Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of kd for UniProtKB: P41594
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395923(CHEMBL2164550)
Affinity DataKd:  2.25nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395923(CHEMBL2164550)
Affinity DataKd:  3.80nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counter in absence of MPEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395923(CHEMBL2164550)
Affinity DataKd:  5.5nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counter in presence of 10 nM MPEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50395923(CHEMBL2164550)
Affinity DataKd:  7.20nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST after 1 hr by scintillation counter in presence of 20 nM MPEPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50084137(2-Methyl-6-(phenylethynyl)pyridine | 2-Methyl-6-ph...)
Affinity DataKd:  8.60nMAssay Description:Binding affinity to human mGluR5 expressed in HEK293 cell membranes expressing GLAST by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed