TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Displacement of [18F]-LU13 from rat spleen CB2 receptor incubated for 90 mins by competitive radioligand binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Agonist activity at rat CB2 receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP production treated 15 mins before fors...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 9.33nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production after 20 mins ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 9.55nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production after 20 mins ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Agonist activity at rat CB2 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP levelMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Agonist activity at rat CB2 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP levelMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Agonist activity at rat CB2 receptor expressed in CHOK1 cells assessed as inhibition of forskolin-induced cAMP production treated 15 mins before fors...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in rat spleen homogenate after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in rat spleen homogenate after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from CB2 receptor in rat spleen homogenate after 90 minsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]WIN-55212-2 from CB2 receptor in Sprague-Dawley rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat cannabinoid CB2 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 1.55E+3nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in HEK293 cells co-expressing chimeric Gaq/o protein by FLIPR assay by FLIPR assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Displacement of [3H]WIN-55212-2 from CB2 receptor in Sprague-Dawley rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of [3H]WIN-55212-2 from CB2 receptor in Sprague-Dawley rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: 4.03E+3nMAssay Description:Displacement of [3H]WIN-55212-2 from CB2 receptor in Sprague-Dawley rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to CB2 receptor in rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to CB2 receptor in rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production after 20 mins ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to CB2 receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to CB2 receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to CB2 receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to CB2 receptor in rat spleen membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Helmholtz-Zentrum Dresden-Rossendorf (Hzdr)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production after 20 mins ...More data for this Ligand-Target Pair