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Report error Found 296 of ic50 for UniProtKB: P14625
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50005782(ATI-13387X | ONALESPIB)
Affinity DataIC50: 22nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataIC50: 26nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087812(CHEMBL3426787)
Affinity DataIC50: 32nMAssay Description:Inhibition of GRP94 (unknown origin) expressed in HEK293 cells assessed as reduction of Toll-like receptor trafficking to cell membrane treated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50439621(STA-9090 | GANETESPIB)
Affinity DataIC50: 38nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540240(CHEMBL4647894)
Affinity DataIC50: 49nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555415(CHEMBL4744238)
Affinity DataIC50: 50nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540237(CHEMBL4647171)
Affinity DataIC50: 54nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540232(CHEMBL4641526)
Affinity DataIC50: 78nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540239(CHEMBL4635982)
Affinity DataIC50: 78nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM20926(5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-N-ethyl-4-...)
Affinity DataIC50: 85nMAssay Description:Inhibition of Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540236(CHEMBL4639163)
Affinity DataIC50: 89nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540249(CHEMBL4635778)
Affinity DataIC50: 96nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540248(CHEMBL4648197)
Affinity DataIC50: 100nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087810(CHEMBL3426784 | US9630965, Compound 52 | US1042806...)
Affinity DataIC50: 101nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165316(8-(2,4-Dichloro-phenylsulfanyl)-9-pent-4-ynyl-9H-p...)
Affinity DataIC50: 120nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataIC50: 132nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165315(9-Pent-4-ynyl-8-(2,4,5-trichloro-phenylsulfanyl)-9...)
Affinity DataIC50: 170nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540242(CHEMBL4648091)
Affinity DataIC50: 175nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540238(CHEMBL4638275)
Affinity DataIC50: 190nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540251(CHEMBL4641450)
Affinity DataIC50: 192nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50571896(CHEMBL4869481)
Affinity DataIC50: 194nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555456(CHEMBL4779990)
Affinity DataIC50: 195nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555451(CHEMBL4782374)
Affinity DataIC50: 196nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540241(CHEMBL4636983)
Affinity DataIC50: 197nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555440(CHEMBL4797602)
Affinity DataIC50: 198nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50169935(CHEMBL3805249)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50540250(CHEMBL4649532)
Affinity DataIC50: 209nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555455(CHEMBL4753741)
Affinity DataIC50: 216nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555442(CHEMBL4777147)
Affinity DataIC50: 217nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087721(CHEMBL3426781)
Affinity DataIC50: 220nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555447(CHEMBL4753836)
Affinity DataIC50: 232nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087447(CHEMBL3426734)
Affinity DataIC50: 240nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555416(CHEMBL4781723)
Affinity DataIC50: 245nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165268(8-(3,5-Dichloro-phenylsulfanyl)-9-pent-4-ynyl-9H-p...)
Affinity DataIC50: 260nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087811(CHEMBL3426785)
Affinity DataIC50: 265nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087454(CHEMBL3426741)
Affinity DataIC50: 287nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087448(CHEMBL3426735)
Affinity DataIC50: 290nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50555441(CHEMBL4744192)
Affinity DataIC50: 290nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50180302(8-[(6-IODO-1,3-BENZODIOXOL-5-YL)THIO]-9-[3-(ISOPRO...)
Affinity DataIC50: 301nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50571903(CHEMBL4863672)
Affinity DataIC50: 318nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087575(CHEMBL3426763)
Affinity DataIC50: 340nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165295(8-(2-Chloro-phenylsulfanyl)-9-pent-4-ynyl-9H-purin...)
Affinity DataIC50: 350nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 350nMAssay Description:Inhibition of HSP90B1 (unknown origin) incubated for 1 hr by colloidal coomassie staining based LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087524(CHEMBL3426756)
Affinity DataIC50: 390nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087445(CHEMBL3426733)
Affinity DataIC50: 390nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087720(CHEMBL3426780)
Affinity DataIC50: 410nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087507(CHEMBL3426748)
Affinity DataIC50: 429nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50087452(CHEMBL3426739)
Affinity DataIC50: 430nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50240873(CHEMBL4068596)
Affinity DataIC50: 448nMAssay Description:Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetEndoplasmin(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50450704(CHEMBL560895 | SNX-2112)
Affinity DataIC50: 484nMAssay Description:Inhibition of recombinant GRP94 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
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