Compile Data Set for Download or QSAR
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TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataKon:  0.360M-1s-1Assay Description:Binding affinity to PPARalpha (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50235985(CHEMBL4092600)
Affinity DataKon:  0.0160M-1s-1Assay Description:Binding affinity to PPARalpha (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50235986(CHEMBL4073499)
Affinity DataKon:  0.0250M-1s-1Assay Description:Binding affinity to PPARalpha (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed