Compile Data Set for Download or QSAR
maximum 50k data
Found 124 of ec50 data for complexid = 50000781,50005864
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50368543(CHEMBL605668)
Affinity DataEC50:  0.191nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50230152(Binodenoson | Corvue | MRE0470 | WRC-0470)
Affinity DataEC50:  0.257nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421975(CHEMBL611607)
Affinity DataEC50:  0.324nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421890(CHEMBL2311197)
Affinity DataEC50:  0.389nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421980(CHEMBL2113592)
Affinity DataEC50:  0.468nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406504(CHEMBL605878)
Affinity DataEC50:  0.501nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421982(CHEMBL608663)
Affinity DataEC50:  0.692nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406519(CHEMBL606080)
Affinity DataEC50:  0.871nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421985(CHEMBL611916)
Affinity DataEC50:  1nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406499(CHEMBL605463)
Affinity DataEC50:  1.40nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406511(CHEMBL604836)
Affinity DataEC50:  1.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421983(CHEMBL608966)
Affinity DataEC50:  1.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406503(CHEMBL606081)
Affinity DataEC50:  1.90nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009509((CGS 22,492) 2-[6-Amino-2-(2-cyclohexyl-ethylamino...)
Affinity DataEC50:  1.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421972(CHEMBL611921)
Affinity DataEC50:  2nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009535((CGS 22,989) 2-[6-Amino-2-(2-cyclohex-1-enyl-ethyl...)
Affinity DataEC50:  2.20nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406518(CHEMBL604422)
Affinity DataEC50:  2.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406510(CHEMBL605876)
Affinity DataEC50:  2.60nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406501(CHEMBL606092)
Affinity DataEC50:  2.80nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421979(CHEMBL607585)
Affinity DataEC50:  2.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406514(CHEMBL605873)
Affinity DataEC50:  3nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421986(CHEMBL610443)
Affinity DataEC50:  3.30nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406521(CHEMBL605461)
Affinity DataEC50:  3.40nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421976(CHEMBL607796)
Affinity DataEC50:  3.5nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406509(CHEMBL605667)
Affinity DataEC50:  3.70nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406506(CHEMBL606305)
Affinity DataEC50:  3.80nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406508(CHEMBL605465)
Affinity DataEC50:  4.90nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406507(CHEMBL604837)
Affinity DataEC50:  5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406512(CHEMBL603587)
Affinity DataEC50:  5.5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421978(CHEMBL611314)
Affinity DataEC50:  5.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406502(CHEMBL604212)
Affinity DataEC50:  6.30nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421971(CHEMBL611917)
Affinity DataEC50:  7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421984(CHEMBL607599)
Affinity DataEC50:  7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406505(CHEMBL605257)
Affinity DataEC50:  9.5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406520(CHEMBL605256)
Affinity DataEC50:  9.80nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421977(CHEMBL609231)
Affinity DataEC50:  13nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406516(CHEMBL605048)
Affinity DataEC50:  22nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50406513(CHEMBL605250)
Affinity DataEC50:  32nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421973(CHEMBL610727)
Affinity DataEC50:  35nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421981(CHEMBL607877)
Affinity DataEC50:  50nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM14487((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataEC50:  51nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50453222(CHEMBL2113509)
Affinity DataEC50:  62nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421889(CHEMBL2311199)
Affinity DataEC50:  62nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421974(CHEMBL607873)
Affinity DataEC50:  76nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50368478(CHEMBL610444)
Affinity DataEC50:  79nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50453224(2-(l-hexyn-l-yl)-adenosine-5'-N-methyluronamide (1...)
Affinity DataEC50:  105nMAssay Description:Inhibition of adenylate cyclase via Adenosine A1 receptor in rat fat cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50389797(CHEMBL261482)
Affinity DataEC50:  110nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50453221(CHEMBL2113510)
Affinity DataEC50:  127nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50119168((2R,3R,4S,5R)-2-(6-Amino-2-hex-1-ynyl-purin-9-yl)-...)
Affinity DataEC50:  128nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  130nMAssay Description:Potency against PC12 cell A2 adenosine receptor by adenylate cyclase activationMore data for this Ligand-Target Pair
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