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Found 3 of ic50 data for complexid = 50000079
TargetCalpain-1/Calpain-2 catalytic subunit(Homo sapiens (Human))
Roche Pharma Research And Early Development

Curated by ChEMBL
LigandPNGBDBM50536838(CHEMBL4520267)
Affinity DataIC50:  96nMAssay Description:Inhibition of calpain (unknown origin) using calpain substrate preincubated for 20 mins followed by substrate addition by fluorescence plate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1/Calpain-2 catalytic subunit(Homo sapiens (Human))
Roche Pharma Research And Early Development

Curated by ChEMBL
LigandPNGBDBM50536839(CHEMBL2402203 | acs.jmedchem.1c00409_ST.724)
Affinity DataIC50:  600nMAssay Description:Inhibition of calpain (unknown origin) using calpain substrate preincubated for 20 mins followed by substrate addition by fluorescence plate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1/Calpain-2 catalytic subunit(Homo sapiens (Human))
Roche Pharma Research And Early Development

Curated by ChEMBL
LigandPNGBDBM50536834(CHEMBL4590201)
Affinity DataIC50:  600nMAssay Description:Inhibition of calpain (unknown origin) using calpain substrate preincubated for 20 mins followed by substrate addition by fluorescence plate reader a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed