Compile Data Set for Download or QSAR
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Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50005112
LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | 3-aminopropylphos...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | 3-aminopropylphos...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24185((3-aminopropyl)(methyl)phosphinic acid | 3-Apmpa |...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
LigandPNGBDBM50032964((R)-4-Amino-3-(4-chloro-phenyl)-butyric acid | 4-A...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
LigandPNGBDBM24185((3-aminopropyl)(methyl)phosphinic acid | 3-Apmpa |...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataIC50:  17nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
LigandPNGBDBM24186((3-amino-2-hydroxypropyl)phosphinic acid | 3-amino...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataIC50:  25nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
LigandPNGBDBM24189(3-aminopropylphosphinic derivative, (R)-4 | 3-amin...)
Affinity DataIC50:  29nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to cat Gamma-aminobutyric acid type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032964((R)-4-Amino-3-(4-chloro-phenyl)-butyric acid | 4-A...)
Affinity DataIC50:  32nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)
Affinity DataIC50:  35nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
LigandPNGBDBM50032958(CHEMBL430501 | [3-Amino-2-(4-chloro-phenyl)-propyl...)
Affinity DataIC50:  39nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24189(3-aminopropylphosphinic derivative, (R)-4 | 3-amin...)
Affinity DataIC50:  45nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24189(3-aminopropylphosphinic derivative, (R)-4 | 3-amin...)
Affinity DataIC50:  45nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032969(CHEMBL321255 | [3-Amino-2-(4-chloro-phenyl)-2-hydr...)
Affinity DataIC50:  65nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032968((3-Amino-propyl)-difluoromethyl-phosphinic acid | ...)
Affinity DataIC50:  89nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)
Affinity DataIC50:  107nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
LigandPNGBDBM50032971((3-Amino-1-methyl-propyl)-methyl-phosphinic acid |...)
Affinity DataIC50:  140nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM24189(3-aminopropylphosphinic derivative, (R)-4 | 3-amin...)
Affinity DataIC50:  152nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032971((3-Amino-1-methyl-propyl)-methyl-phosphinic acid |...)
Affinity DataIC50:  166nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to cat Gamma-aminobutyric acid type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032961((3-Amino-2-hydroxy-propyl)-difluoromethyl-phosphin...)
Affinity DataIC50:  213nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataIC50:  280nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032959(CHEMBL111378 | [3-Amino-2-(4-fluoro-phenyl)-propyl...)
Affinity DataIC50:  360nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032970((3-Amino-butyl)-phosphinic acid | CHEMBL113907)
Affinity DataIC50:  500nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataIC50:  665nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032975((3-Amino-2-methyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataIC50:  780nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032977((3-Amino-2-phenyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataIC50:  880nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032967((3-Amino-1-methyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataIC50:  920nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032979((3-Amino-propyl)-hydroxymethyl-phosphinic acid | C...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032966((3-Amino-1-hydroxy-propyl)-methyl-phosphinic acid ...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032972((3-Amino-propyl)-ethyl-phosphinic acid | CGP-36216...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032963((S)-4-Amino-3-(4-chloro-phenyl)-butyric acid | BAC...)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032972((3-Amino-propyl)-ethyl-phosphinic acid | CGP-36216...)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataIC50:  4.41E+3nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032981((3-Amino-propyl)-phosphonic acid | CHEMBL286077 | ...)
Affinity DataIC50:  6.81E+3nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032965(((R)-3-Amino-2-hydroxy-butyl)-phosphinic acid | CH...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032974((3-Amino-1-ethyl-propyl)-methyl-phosphinic acid | ...)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50032960((3-Amino-1-trifluoromethyl-propyl)-methyl-phosphin...)
Affinity DataIC50:  6.76E+4nMAssay Description:Inhibition of [3H]-CGP-27,492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed