Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50005113
LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | 3-aminopropylphos...)
Affinity DataIC50:  5nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM24185((3-aminopropyl)(methyl)phosphinic acid | 3-Apmpa |...)
Affinity DataIC50:  16nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

LigandPNGBDBM50033007((3-Amino-propyl)-(3-oxo-butyl)-phosphinic acid | C...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033008((3-Amino-propyl)-[3-(2-carbamoyl-benzoylamino)-2-h...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032996((3-Amino-propyl)-[2-(tetrahydro-pyran-2-yl)-ethyl]...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033024((3-Amino-propyl)-(2-cyclohexyl-ethyl)-phosphinic a...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032972((3-Amino-propyl)-ethyl-phosphinic acid | CGP-36216...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033017((3-Amino-propyl)-cyclohexylmethyl-phosphinic acid ...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032989(((S)-3-Amino-2-hydroxy-propyl)-cyclohexylmethyl-ph...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032989(((S)-3-Amino-2-hydroxy-propyl)-cyclohexylmethyl-ph...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032987((3-Amino-propyl)-pyridin-2-ylmethyl-phosphinic aci...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032984(CHEMBL113305 | [3-Amino-2-(4-chloro-phenyl)-2-hydr...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032989(((S)-3-Amino-2-hydroxy-propyl)-cyclohexylmethyl-ph...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033004(CHEMBL321688 | [3-Amino-2-(4-chloro-phenyl)-2-hydr...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033016((3-Amino-propyl)-(hydroxy-phenyl-methyl)-phosphini...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033011(CHEMBL114128 | [3-Amino-2-(4-chloro-phenyl)-propyl...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033029((3-Amino-propyl)-phenethyl-phosphinic acid | CHEMB...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033018((3-Amino-propyl)-benzyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032997(((S)-3-Amino-2-hydroxy-propyl)-diethoxymethyl-phos...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032995((3-Amino-2-oxo-propyl)-cyclopropylmethyl-phosphini...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032990((3-Amino-propyl)-isobutyl-phosphinic acid | CHEMBL...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032997(((S)-3-Amino-2-hydroxy-propyl)-diethoxymethyl-phos...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033013((3-Amino-propyl)-propyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033019((3-Amino-propyl)-diisopropoxymethyl-phosphinic aci...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032994((3-Amino-propyl)-(1-hydroxy-butyl)-phosphinic acid...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033027((3-Amino-propyl)-hexyl-phosphinic acid | CHEMBL113...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033021((3-Amino-propyl)-dibutoxymethyl-phosphinic acid | ...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033009(CHEMBL114812 | [3-Amino-2-(4-chloro-phenyl)-propyl...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033012((3-Amino-propyl)-(1,1-difluoro-butyl)-phosphinic a...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033003((3-Amino-propyl)-diethoxymethyl-phosphinic acid | ...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

LigandPNGBDBM50032986((3-Amino-propyl)-dipropoxymethyl-phosphinic acid |...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032985(Bis-(3-amino-propyl)-phosphinic acid | CHEMBL11229...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032998((3-Amino-2-hydroxy-propyl)-butyl-phosphinic acid |...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033000((3-Amino-propyl)-(tetrahydro-pyran-2-ylmethyl)-pho...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033014(((R)-3-Amino-2-hydroxy-propyl)-benzyl-phosphinic a...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032992((3-Amino-propyl)-(tetrahydro-furan-2-yl)-phosphini...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033028((3-Amino-1-hydroxy-propyl)-butyl-phosphinic acid |...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033001((3-Amino-propyl)-cyclopropylmethyl-phosphinic acid...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032982((3-Amino-propyl)-butyl-phosphinic acid | 3-aminopr...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033026((3-Amino-propyl)-(tetrahydro-pyran-2-yl)-phosphini...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032983((3-Amino-2-hydroxy-2-methyl-propyl)-butyl-phosphin...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033023(Aminomethyl-(3-amino-propyl)-phosphinic acid | CHE...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033025((3-Amino-2-oxo-propyl)-cyclohexylmethyl-phosphinic...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033002((3-Amino-propyl)-(4-fluoro-benzyl)-phosphinic acid...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50033010((3-Amino-propyl)-tert-butyl-phosphinic acid | CHEM...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032993((3-Amino-propyl)-phenyl-phosphinic acid | CHEMBL11...)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50032988((3-Amino-1-methyl-propyl)-butyl-phosphinic acid | ...)
Affinity DataIC50:  3.41E+5nMAssay Description:Inhibition of binding of [3H]-CGP-27,492 to gamma-aminobutyric acid type B receptor of rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed