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Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50018486
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196343(2,2-Dimethyl-propionic acid 2-(4-tert-butyl-benzyl...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196366(2-((3-(2-chloro-4-hydroxy-5-methoxybenzyl)thiourei...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196365(2-((3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196341(2-((3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196365(2-((3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  13.3nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196337(2,2-Dimethyl-propionic acid 2-(3,4-dimethyl-benzyl...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196354(2-((3-(3-bromo-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196336(2-((3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196367(2-((3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196352(2-((3-(3-chloro-4-hydroxy-5-methoxybenzyl)thiourei...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196336(2-((3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  23nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196357(2-((3-(2-chloro-4-hydroxy-5-methoxybenzyl)thiourei...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196335(2-(3-(3-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196350(1-(2-bromo-4-hydroxy-5-methoxybenzyl)-3-(4-tert-bu...)
Affinity DataKi:  30nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196355(2-((3-(3-chloro-4-hydroxy-5-methoxybenzyl)thiourei...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196327(2-((3-(3-bromo-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196346(2-(3-(4-hydroxy-3-methoxybenzyl)thioureido)-3-(4-t...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196364(1-(2-chloro-4-hydroxy-5-methoxybenzyl)-3-(4-tert-b...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196348(2-(3-(4-hydroxy-3-methoxybenzyl)thioureido)-4-(4-t...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196360(2-(3-(3-bromo-4-hydroxy-5-methoxybenzyl)thioureido...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196356(2-(3-(4-hydroxy-3-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196350(1-(2-bromo-4-hydroxy-5-methoxybenzyl)-3-(4-tert-bu...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196362(2-(3-(2-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196358(2-((3-(4-hydroxy-3-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196340(1-(3-bromo-4-hydroxy-5-methoxybenzyl)-3-(4-tert-bu...)
Affinity DataKi:  49nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196340(1-(3-bromo-4-hydroxy-5-methoxybenzyl)-3-(4-tert-bu...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196341(2-((3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  55nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196334(2-(3-(4-hydroxy-3-methoxybenzyl)thioureido)-4-(3,4...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196351(1-(4-tert-Butyl-benzyl)-3-(4-hydroxy-3-methoxy-ben...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196342(2-(3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  69nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196329(2-(3-(2-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  72nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196361(2-(3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureido...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196331(2-(3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureido...)
Affinity DataKi:  75nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196331(2-(3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureido...)
Affinity DataKi:  76nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196363(1-(3-chloro-4-hydroxy-5-methoxybenzyl)-3-(4-tert-b...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196342(2-(3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196329(2-(3-(2-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196333(2-(3-(3-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196347(2-(3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196339(2-(3-(3-bromo-4-hydroxy-5-methoxybenzyl)thioureido...)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196358(2-((3-(4-hydroxy-3-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  103nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196368(2-(3-(2-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196359(2-(3-(2-bromo-4-hydroxy-5-methoxybenzyl)thioureido...)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196353(2-(3-(4-hydroxy-3-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  115nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196332(2-((3-(4-hydroxy-3-iodo-5-methoxybenzyl)thioureido...)
Affinity DataKi:  121nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196344(2-(3-(3-chloro-4-hydroxy-5-methoxybenzyl)thioureid...)
Affinity DataKi:  122nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50170053(CHEMBL177809 | N-(4-hydroxy-2-iodo-5-methoxybenzyl...)
Affinity DataKi:  127nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of calcium uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196353(2-(3-(4-hydroxy-3-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196330(1-(4-tert-butylbenzyl)-3-(4-hydroxy-2-iodo-5-metho...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196338(2-(3-(4-hydroxy-2-iodo-5-methoxybenzyl)thioureido)...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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