Compile Data Set for Download or QSAR
Found 44 Enz. Inhib. hit(s) with all data for entry = 50008591
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075089(CHEMBL133420 | Sodium; [2-(4-chloro-benzenesulfony...)
Affinity DataIC50:  2.20nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075088(CHEMBL336846 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075086(CHEMBL341221 | Sodium; [2-(benzenesulfonylamino-me...)
Affinity DataIC50:  13nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075091(CHEMBL131894 | Sodium; 3-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  15nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075077(CHEMBL131497 | Sodium; {2-[(naphthalene-2-sulfonyl...)
Affinity DataIC50:  22nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075082(CHEMBL264516 | Sodium; 2-[(4-chloro-benzenesulfony...)
Affinity DataIC50:  26nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075094(CHEMBL132659 | Sodium; {2-[2-(4-chloro-benzenesulf...)
Affinity DataIC50:  32nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075093(CHEMBL130377 | Sodium; 5-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  36nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50002805((daltroban){4-[2-(4-Chloro-benzenesulfonylamino)-e...)
Affinity DataIC50:  37nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075079(CHEMBL334501 | Sodium; 4-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  39nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075096(CHEMBL336352 | Sodium; 2-[2-(4-chloro-benzenesulfo...)
Affinity DataIC50:  66nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075076(CHEMBL335043 | Sodium; {2-[(thiophene-2-sulfonylam...)
Affinity DataIC50:  85nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075092(CHEMBL339994 | Sodium; 2-[3-(4-chloro-benzenesulfo...)
Affinity DataIC50:  85nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075085(CHEMBL131036 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  141nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075091(CHEMBL131894 | Sodium; 3-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  160nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075090(CHEMBL422441 | Sodium; {2-[(naphthalene-1-sulfonyl...)
Affinity DataIC50:  295nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075085(CHEMBL131036 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  320nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075089(CHEMBL133420 | Sodium; [2-(4-chloro-benzenesulfony...)
Affinity DataIC50:  360nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075088(CHEMBL336846 | Sodium; {2-[(4-chloro-benzenesulfon...)
Affinity DataIC50:  360nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50002805((daltroban){4-[2-(4-Chloro-benzenesulfonylamino)-e...)
Affinity DataIC50:  460nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075081(CHEMBL130045 | Sodium; 2-[4-(4-chloro-benzenesulfo...)
Affinity DataIC50: >479nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075084(CHEMBL130170 | Sodium; {2-[3-(4-chloro-benzenesulf...)
Affinity DataIC50:  513nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075077(CHEMBL131497 | Sodium; {2-[(naphthalene-2-sulfonyl...)
Affinity DataIC50:  950nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075095(CHEMBL131336 | Sodium; {2-[4-(4-chloro-benzenesulf...)
Affinity DataIC50:  977nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075086(CHEMBL341221 | Sodium; [2-(benzenesulfonylamino-me...)
Affinity DataIC50:  1.02E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075080(CHEMBL130460 | Sodium; [2-(cyclohexanesulfonylamin...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075082(CHEMBL264516 | Sodium; 2-[(4-chloro-benzenesulfony...)
Affinity DataIC50:  1.32E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075079(CHEMBL334501 | Sodium; 4-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  1.34E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075083(CHEMBL340073 | Sodium; {2-[(pentane-1-sulfonylamin...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075094(CHEMBL132659 | Sodium; {2-[2-(4-chloro-benzenesulf...)
Affinity DataIC50:  1.48E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075087(CHEMBL134128 | Sodium; {2-[(pyridine-3-sulfonylami...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075076(CHEMBL335043 | Sodium; {2-[(thiophene-2-sulfonylam...)
Affinity DataIC50:  2.81E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075093(CHEMBL130377 | Sodium; 5-{2-[(4-chloro-benzenesulf...)
Affinity DataIC50:  2.88E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(RAT)
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075078(CHEMBL132573 | Sodium; [2-(phenylmethanesulfonylam...)
Affinity DataIC50:  5.90E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075092(CHEMBL339994 | Sodium; 2-[3-(4-chloro-benzenesulfo...)
Affinity DataIC50:  6.60E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075096(CHEMBL336352 | Sodium; 2-[2-(4-chloro-benzenesulfo...)
Affinity DataIC50:  7.76E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075080(CHEMBL130460 | Sodium; [2-(cyclohexanesulfonylamin...)
Affinity DataIC50:  1.78E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075090(CHEMBL422441 | Sodium; {2-[(naphthalene-1-sulfonyl...)
Affinity DataIC50:  4.79E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075084(CHEMBL130170 | Sodium; {2-[3-(4-chloro-benzenesulf...)
Affinity DataIC50:  7.23E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075083(CHEMBL340073 | Sodium; {2-[(pentane-1-sulfonylamin...)
Affinity DataIC50:  7.76E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075087(CHEMBL134128 | Sodium; {2-[(pyridine-3-sulfonylami...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075095(CHEMBL131336 | Sodium; {2-[4-(4-chloro-benzenesulf...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075081(CHEMBL130045 | Sodium; 2-[4-(4-chloro-benzenesulfo...)
Affinity DataIC50:  1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Zeria Pharmaceutical Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50075078(CHEMBL132573 | Sodium; [2-(phenylmethanesulfonylam...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed