Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50020836
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218188((R)-2-(2-(4-(oxazol-5-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218175((R)-N-(5-(2-(4-(2-ethylthiazol-4-yl)phenethylamino...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218174((R)-2-(2-(4-(2-phenylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataEC50:  580nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218172((R)-2-(2-(4-(2-cyclopentylthiazol-4-yl)phenoxy)eth...)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218178((1R)-2-(4-(2-(pyridin-3-yl)thiazol-4-yl)phenethyla...)
Affinity DataEC50:  1.19E+3nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218181((R)-2-(2-(4-(5-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataEC50:  309nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218173((R)-2-(2-(4-(2-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218176((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-4-yl)thia...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218187((R)-N-(5-(2-(4-(2-phenylthiazol-4-yl)phenethylamin...)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218186((R)-2-(4-(2-phenylthiazol-4-yl)phenethylamino)-1-(...)
Affinity DataEC50:  2.74E+3nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218184((R)-N-(5-(2-(4-(2-methylthiazol-4-yl)phenethylamin...)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218167((R)-2-(2-(4-(2-isopropyloxazol-4-yl)phenoxy)ethyla...)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218177((R)-2-(2-(4-(2-(benzyloxymethyl)oxazol-4-yl)phenox...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218166((R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218182((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(trifluoromethyl)t...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218183((R)-2-(4-(2-methylthiazol-4-yl)phenethylamino)-1-(...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218163((R)-2-(2-(4-(oxazol-2-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataEC50:  520nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat adrenergic beta-3 receptor assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218185((1R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-3-yl)thi...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218189((R)-2-(4-(2-ethylthiazol-4-yl)phenethylamino)-1-(p...)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50092645(N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at rat adrenergic beta-3 receptor assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218170((R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218169((R)-2-(4-(2-(trifluoromethyl)thiazol-4-yl)phenethy...)
Affinity DataEC50:  4.49E+3nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218168((R)-2-(2-(4-(2-ethyloxazol-4-yl)phenoxy)ethylamino...)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218180((R)-2-(2-(4-(2-ethylthiazol-4-yl)phenoxy)ethylamin...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218179((R)-2-(2-(4-(2,5-dimethyloxazol-4-yl)phenoxy)ethyl...)
Affinity DataEC50:  606nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218171((R)-2-(2-(4-(2-(methoxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataEC50:  47nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218166((R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218173((R)-2-(2-(4-(2-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218170((R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218180((R)-2-(2-(4-(2-ethylthiazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218168((R)-2-(2-(4-(2-ethyloxazol-4-yl)phenoxy)ethylamino...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218167((R)-2-(2-(4-(2-isopropyloxazol-4-yl)phenoxy)ethyla...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218177((R)-2-(2-(4-(2-(benzyloxymethyl)oxazol-4-yl)phenox...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218176((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-4-yl)thia...)
Affinity DataKi:  97nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218182((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(trifluoromethyl)t...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218185((1R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-3-yl)thi...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218172((R)-2-(2-(4-(2-cyclopentylthiazol-4-yl)phenoxy)eth...)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218174((R)-2-(2-(4-(2-phenylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218181((R)-2-(2-(4-(5-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218166((R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218171((R)-2-(2-(4-(2-(methoxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50218170((R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataKi:  270nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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