Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50028470
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257185((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257186((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-azido...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  1.05nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  1.64nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240844((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-aceta...)
Affinity DataKi:  1.81nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257188((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataKi:  2.01nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257194((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-(7-aminoheptanam...)
Affinity DataKi:  2.99nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257192((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-a...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257187((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino...)
Affinity DataKi:  4.87nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257192((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-a...)
Affinity DataKi:  5.49nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257189((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataKi:  8.07nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257193((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataKi:  9.90nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257193((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataKi:  10.4nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257191((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-(...)
Affinity DataKi:  20.3nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240339((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-5-g...)
Affinity DataKi:  95nMAssay Description:Binding affinity to human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257197((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataKi:  105nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257190((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3-acetamido...)
Affinity DataKi:  136nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240339((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-5-g...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257195((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataKi:  303nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257199((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-(5-guani...)
Affinity DataKi:  631nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257196((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-2-acetamido...)
Affinity DataKi:  647nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257198((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataKi:  2.17E+3nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257185((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataIC50:  0.383nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257186((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-azido...)
Affinity DataIC50:  0.970nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50248034(2-{[1-(7-Chloro-quinolin-4-yl)-5-(2,6-dimethoxy-ph...)
Affinity DataIC50:  0.990nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataIC50:  2.19nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240844((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-aceta...)
Affinity DataIC50:  2.42nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257188((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataIC50:  2.68nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257194((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-(7-aminoheptanam...)
Affinity DataIC50:  3.99nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257187((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino...)
Affinity DataIC50:  6.5nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257192((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-a...)
Affinity DataIC50:  7.32nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257189((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataIC50:  10.8nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257193((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataIC50:  13.9nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257191((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-7-amino-3-(...)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257197((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257190((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3-acetamido...)
Affinity DataIC50:  181nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240339((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-5-g...)
Affinity DataIC50:  240nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257195((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataIC50:  403nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257199((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-(5-guani...)
Affinity DataIC50:  842nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257196((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-2-acetamido...)
Affinity DataIC50:  863nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257198((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataIC50:  2.90E+3nMAssay Description:Displacement of [125I]I-Tyr(3)NT from human NTR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataEC50:  1.98nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257189((S)-2-((S)-2-((S)-2-((S)-1-((S)-2-((S)-3,7-diamino...)
Affinity DataEC50:  6.21nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257187((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino...)
Affinity DataEC50:  7.76nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257188((S)-2-((2S,3R)-2-((S)-2-((S)-1-((S)-5-guanidino-2-...)
Affinity DataEC50:  1.85nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257199((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-(5-guani...)
Affinity DataEC50:  783nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50257198((S)-2-((S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2-a...)
Affinity DataEC50:  1.86E+3nMAssay Description:Agonist activity at NTR1 in human HT-29 cells assessed as increase in intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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