Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50048335
LigandChemical structure of BindingDB Monomer ID 50056419BDBM50056419(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  0.251nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor was determined in rat cerebro cortical membranes using [3H]quipazine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212854BDBM50212854(CHEMBL283483)
Affinity DataKi:  0.794nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor was determined in rat cerebro cortical membranes using [3H]quipazine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50031475BDBM50031475(4-Amino-N-(R)-1-aza-bicyclo[2.2.2]oct-3-yl-5-chlor...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor was determined in rat cerebro cortical membranes using [3H]quipazine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 85330BDBM85330(NSC_68647 | CAS_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor was determined in rat cerebro cortical membranes using [3H]quipazine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 10755BDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | CHEMBL535832 | ...)
Affinity DataEC50:  6.30nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212855BDBM50212855(CHEMBL28499)
Affinity DataKi:  10nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor was determined in rat cerebro cortical membranes using [3H]quipazine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212855BDBM50212855(CHEMBL28499)
Affinity DataEC50:  13nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212856BDBM50212856(CHEMBL27966)
Affinity DataEC50:  32nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212856BDBM50212856(CHEMBL27966)
Affinity DataKi:  40nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor was determined in rat cerebro cortical membranes using [3H]quipazine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50056419BDBM50056419(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataEC50:  63nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50031475BDBM50031475(4-Amino-N-(R)-1-aza-bicyclo[2.2.2]oct-3-yl-5-chlor...)
Affinity DataEC50:  501nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50212854BDBM50212854(CHEMBL283483)
Affinity DataEC50: <1.00E+3nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity in the rat esophageal muscularis mucosaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/20/2018
Entry Details