Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50048490
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50218267(CHEMBL74404)
Affinity DataIC50: 10nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218268(CHEMBL309341)
Affinity DataIC50: 19nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218265(CHEMBL308407)
Affinity DataIC50: 30nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218263(CHEMBL419814)
Affinity DataIC50: 30nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218262(CHEMBL308158)
Affinity DataIC50: 39nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218264(CHEMBL72362)
Affinity DataIC50: 42nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218260(CHEMBL70391)
Affinity DataIC50: 53nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218261(CHEMBL74631)
Affinity DataIC50: 57nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50092350((5-Cyclopentyloxy-6-methoxy-phthalazin-1-yl)-(3,5-...)
Affinity DataIC50: 59nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218269(CHEMBL73640)
Affinity DataIC50: 153nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218266(CHEMBL303880)
Affinity DataIC50: 186nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50218261(CHEMBL74631)
Affinity DataKi:  13nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218265(CHEMBL308407)
Affinity DataKi:  16nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218262(CHEMBL308158)
Affinity DataKi:  46nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218267(CHEMBL74404)
Affinity DataKi:  71nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50092350((5-Cyclopentyloxy-6-methoxy-phthalazin-1-yl)-(3,5-...)
Affinity DataKi:  95nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218264(CHEMBL72362)
Affinity DataKi:  121nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218260(CHEMBL70391)
Affinity DataKi:  149nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218268(CHEMBL309341)
Affinity DataKi:  164nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218269(CHEMBL73640)
Affinity DataKi:  286nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50218263(CHEMBL419814)
Affinity DataKi:  320nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed