Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50036238
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453355(CHEMBL2113408)
Affinity DataEC50:  6.05E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453348(CHEMBL2113486)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453352(CHEMBL2113416)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453358(CHEMBL2113399)
Affinity DataEC50:  2.43E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453367(CHEMBL2113402)
Affinity DataEC50:  2.37E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453350(CHEMBL2113482)
Affinity DataEC50:  332nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453349(CHEMBL2113483)
Affinity DataEC50:  84nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453362(CHEMBL2113403)
Affinity DataEC50:  730nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453356(CHEMBL2113405)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453224(CHEMBL410873 | 2-(l-hexyn-l-yl)-adenosine-5'-N-met...)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  55nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453353(CHEMBL2113407)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453351(CHEMBL2113485)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453357(CHEMBL2113419)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataEC50:  8.20nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453347(CHEMBL2094083)
Affinity DataEC50:  110nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453365(CHEMBL2113404)
Affinity DataEC50:  475nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453364(CHEMBL2113413)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453346(CHEMBL2113449)
Affinity DataEC50:  167nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453359(CHEMBL2113409)
Affinity DataEC50:  153nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453363(CHEMBL2113412)
Affinity DataEC50:  2.52E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453361(CHEMBL2113411)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453366(CHEMBL2113414)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453354(CHEMBL2113417)
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453360(CHEMBL2113410)
Affinity DataEC50:  657nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  1.30nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453347(CHEMBL2094083)
Affinity DataKi:  2.5nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453356(CHEMBL2113405)
Affinity DataKi:  3nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453365(CHEMBL2113404)
Affinity DataKi:  4nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  10nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453360(CHEMBL2113410)
Affinity DataKi:  11nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453349(CHEMBL2113483)
Affinity DataKi:  14nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453359(CHEMBL2113409)
Affinity DataKi:  20nMAssay Description:Affinity for A1 Adenosine receptor in rat brain using [3H]CHAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453350(CHEMBL2113482)
Affinity DataKi:  28nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453358(CHEMBL2113399)
Affinity DataKi:  33nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453346(CHEMBL2113449)
Affinity DataKi:  35nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453363(CHEMBL2113412)
Affinity DataKi:  38nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453353(CHEMBL2113407)
Affinity DataKi:  42nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453366(CHEMBL2113414)
Affinity DataKi:  47nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453362(CHEMBL2113403)
Affinity DataKi:  49nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453355(CHEMBL2113408)
Affinity DataKi:  70nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453364(CHEMBL2113413)
Affinity DataKi:  100nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453224(CHEMBL410873 | 2-(l-hexyn-l-yl)-adenosine-5'-N-met...)
Affinity DataKi:  130nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453354(CHEMBL2113417)
Affinity DataKi:  167nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453367(CHEMBL2113402)
Affinity DataKi:  184nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453361(CHEMBL2113411)
Affinity DataKi:  236nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453357(CHEMBL2113419)
Affinity DataKi:  267nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453348(CHEMBL2113486)
Affinity DataKi:  398nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453351(CHEMBL2113485)
Affinity DataKi:  656nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50453352(CHEMBL2113416)
Affinity DataKi:  3.30E+3nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed