Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50036909
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086013(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086033(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086017(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086004(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086032(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086029(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086020(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086028(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086001(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086005(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086011(Cyclopropanecarboxylic acid [2-(2-methoxy-6H-isoin...)
Affinity DataKi:  0.950nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086025(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  1.41nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086033(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  1.82nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086015(N-[2-(5,6-Dihydro-indolo[2,1-a]isoquinolin-12-yl)-...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086029(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  4.07nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086032(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  4.37nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086013(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  4.47nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086021(N-[2-(11-Chloro-6,7-dihydro-5H-benzo[3,4]azepino[1...)
Affinity DataKi:  5.01nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086026(Cyclopropanecarboxylic acid [2-(2-ethoxy-6H-isoind...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086017(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  5.89nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086022(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  6.31nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086014(N-[2-(11-Ethoxy-6,7-dihydro-5H-benzo[3,4]azepino[1...)
Affinity DataKi:  6.46nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086005(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  7.24nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086004(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  8.91nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086008(N-[2-(5,6-Dihydro-indolo[2,1-a]isoquinolin-12-yl)-...)
Affinity DataKi:  9.33nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086035(Cyclopropanecarboxylic acid [2-(11-methoxy-6,7-dih...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086010(N-[2-(6H-Isoindolo[2,1-a]indol-11-yl)-ethyl]-butyr...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086028(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  14.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086019(N-[2-(6H-Isoindolo[2,1-a]indol-11-yl)-ethyl]-aceta...)
Affinity DataKi:  17nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086009(N-[2-(6H-Isoindolo[2,1-a]indol-11-yl)-ethyl]-propi...)
Affinity DataKi:  17.4nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086020(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  18.2nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086000(N-[2-(11-Ethoxy-6,7-dihydro-5H-benzo[3,4]azepino[1...)
Affinity DataKi:  21.9nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086007(Cyclobutanecarboxylic acid [2-(11-methoxy-6,7-dihy...)
Affinity DataKi:  31.6nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086034(N-[2-(2-Chloro-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  33.9nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086036(N-[2-(5,6-Dihydro-indolo[2,1-a]isoquinolin-12-yl)-...)
Affinity DataKi:  36.3nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM85065(CAS_117946-91-5 | NSC_122162 | Luzindole)
Affinity DataKi:  44.7nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086003(N-[2-(6,7-Dihydro-5H-benzo[3,4]azepino[1,2-a]indol...)
Affinity DataKi:  45.7nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086011(Cyclopropanecarboxylic acid [2-(2-methoxy-6H-isoin...)
Affinity DataKi:  46.8nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086025(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  52.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086018(Cyclopropanecarboxylic acid [2-(6,7-dihydro-5H-ben...)
Affinity DataKi:  52.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086024(N-[2-(6,7-Dihydro-5H-benzo[3,4]azepino[1,2-a]indol...)
Affinity DataKi:  63.1nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086001(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  66.1nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086015(N-[2-(5,6-Dihydro-indolo[2,1-a]isoquinolin-12-yl)-...)
Affinity DataKi:  70.8nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086024(N-[2-(6,7-Dihydro-5H-benzo[3,4]azepino[1,2-a]indol...)
Affinity DataKi:  79.4nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086030(Cyclopropanecarboxylic acid [2-(11-ethoxy-6,7-dihy...)
Affinity DataKi:  85.1nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086003(N-[2-(6,7-Dihydro-5H-benzo[3,4]azepino[1,2-a]indol...)
Affinity DataKi:  115nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086016(N-[2-(11-Ethoxy-6,7-dihydro-5H-benzo[3,4]azepino[1...)
Affinity DataKi:  117nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086018(Cyclopropanecarboxylic acid [2-(6,7-dihydro-5H-ben...)
Affinity DataKi:  117nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
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