Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50038688
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263386(CHEMBL443967 | H-Arg-N-Me-Arg-Pro-Tyr-Ile-Leu-OH)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263388(CHEMBL507382 | H-Arg-Arg-Pro-Tyr-Ile-Aac-OH)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263387(CHEMBL503059 | H-Arg-Arg-Pro-Tyr-N-Me-Ile-Leu-OH)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50263385(CHEMBL508130 | H-Arg-Arg-Pro-Tyr-Ile-N-Me-Leu-OH)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKd:  0.630nMAssay Description:Displacement of [3H]NT(8-13) from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Human)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50248034(2-{[1-(7-Chloro-quinolin-4-yl)-5-(2,6-dimethoxy-ph...)
Affinity DataKd:  8.90nMAssay Description:Displacement of [3H]SR48692 from wild type human NTR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair