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Found 24 Enz. Inhib. hit(s) with all data for entry = 50039559
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380022(CHEMBL2012509)
Affinity DataIC50:  4.60nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380014(CHEMBL2012500)
Affinity DataIC50:  6.40nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380018(CHEMBL2012505)
Affinity DataIC50:  8.10nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380023(CHEMBL2012510)
Affinity DataIC50:  8.60nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380004(CHEMBL2012489)
Affinity DataIC50:  8.80nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380012(CHEMBL2012497)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380006(CHEMBL2012491)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380019(CHEMBL2012506)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380017(CHEMBL2012503)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380009(CHEMBL2012494)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380011(CHEMBL2012496)
Affinity DataIC50:  21nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380005(CHEMBL2012490)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380003(CHEMBL2012488)
Affinity DataIC50:  24nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380007(CHEMBL2012492)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380013(CHEMBL2012499)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380008(CHEMBL2012493)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380015(CHEMBL2012501)
Affinity DataIC50:  33nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380016(CHEMBL2012502)
Affinity DataIC50:  35nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380010(CHEMBL2012495)
Affinity DataIC50:  45nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380021(CHEMBL2012508)
Affinity DataIC50:  49nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380024(CHEMBL2012511)
Affinity DataIC50:  64nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380002(CHEMBL2012487)
Affinity DataIC50:  225nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380020(CHEMBL2012507)
Affinity DataIC50:  451nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50380001(CHEMBL2012498)
Affinity DataIC50:  513nMAssay Description:Displacement of [3H]haTRAP from human PAR1 after 1 hr by TopCount scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed