Found 30 Enz. Inhib. hit(s) with all data for entry = 50040949 
Affinity DataKi: 1.43nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.82nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.24nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.82nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.84nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.92nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.58nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.89nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11.1nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13.2nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23.4nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 27.2nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 29.1nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 30.3nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53.6nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 75.3nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 90.7nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 97.6nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 99.7nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 165nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 278nMAssay Description:Displacement of [3H]-LSD from cloned human 5HT6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 135nMAssay Description:Antagonist activity at recombinant human 5HT6 receptor expressed in CHO cells assessed as inhibition of 5HT-stimulated cAMP accumulation after 4 hrs ...More data for this Ligand-Target Pair
Affinity DataIC50: 234nMAssay Description:Antagonist activity at recombinant human 5HT6 receptor expressed in CHO cells assessed as inhibition of 5HT-stimulated cAMP accumulation after 4 hrs ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 3.05E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate after 5 mins in presence of NADPHMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate after 5 mins in presence of NADPHMore data for this Ligand-Target Pair
