Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50020462
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630076(CHEMBL5439741)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630094(CHEBI:66437 | Schweinfurthin G | SCHWEINFURTHIN G)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630093(CHEBI:66352 | Vedelianin | VEDELIANIN)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630092(CHEBI:66435 | Schweinfurthin E | SCHWEINFURTHIN E)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630083(CHEMBL5402401)
Affinity DataKi: <1nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630095(CHEBI:66436 | Schweinfurthin F | SCHWEINFURTHIN F)
Affinity DataKi:  6nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630078(CHEMBL5418635)
Affinity DataKi:  16nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630089(CHEMBL5397075)
Affinity DataKi:  31nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630090(CHEMBL5401329)
Affinity DataKi:  37nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630088(CHEMBL5416867)
Affinity DataKi:  43nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630075(CHEMBL5414636)
Affinity DataKi:  46nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630080(CHEMBL5433096)
Affinity DataKi:  64nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630084(CHEMBL5394654)
Affinity DataKi:  119nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630087(CHEMBL5417439)
Affinity DataKi:  254nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630086(CHEBI:66438 | Schweinfurthin H | SCHWEINFURTHIN H)
Affinity DataKi:  401nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630081(CHEMBL5409120)
Affinity DataKi:  523nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630082(CHEMBL5433829)
Affinity DataKi:  829nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630085(CHEMBL5399392)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630091(Mappain | MAPPAIN)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630079(CHEMBL5396667)
Affinity DataKi:  3.22E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetOxysterol-binding protein 1(Homo sapiens)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50630077(CHEMBL5397623)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human C-terminal 6-His tagged OSBP ORD domain (401 to 807 residues) expressed in baculovirus-infected Sf9 cells assessed as reduction i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed