Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50001359
TargetAmyloid-beta precursor protein(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM8963(N-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by thioflavin T-based fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277161(CHEMBL4166095)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by thioflavin T-based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277164(CHEMBL4175715)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by thioflavin T-based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277161(CHEMBL4166095)
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of GSK3beta (unknown origin) using GSM substrate after 30 mins by Kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50214744(Ferulic acid (M5) | ferulic acid | CHEMBL32749 | (...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by thioflavin T-based fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50146456((2E)-3-(3-hydroxyphenyl)prop-2-enoic acid | trans-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by thioflavin T-based fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50237134(CHEMBL1517429)
Affinity DataIC50: 2.66E+5nMAssay Description:Inhibition recombinant human TG2 using N-CbzGlu(gamma-p-nitrophenylester)Gly as substrate after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277163(CHEMBL4177374)
Affinity DataIC50: 4.84E+5nMAssay Description:Inhibition recombinant human TG2 using N-CbzGlu(gamma-p-nitrophenylester)Gly as substrate after 10 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277165(CHEMBL4169514)
Affinity DataIC50: 6.88E+5nMAssay Description:Inhibition recombinant human TG2 using N-CbzGlu(gamma-p-nitrophenylester)Gly as substrate after 10 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277162(CHEMBL4174015)
Affinity DataIC50: 2.00E+6nMAssay Description:Inhibition recombinant human TG2 using N-CbzGlu(gamma-p-nitrophenylester)Gly as substrate after 10 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Alma Mater Studiorum-University of Bologna

Curated by ChEMBL
LigandPNGBDBM50277161(CHEMBL4166095)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition recombinant human TG2 using N-CbzGlu(gamma-p-nitrophenylester)Gly as substrate after 10 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed