Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50001935
Affinity DataKd: 520nMAssay Description:Inhibition of FITC-geldanamycin binding to canine GRP94 incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.38E+3nMAssay Description:Inhibition of FITC-geldanamycin binding to canine GRP94 incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 870nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKd: 200nMAssay Description:Displacement of [3H]NECA from GRP94 in porcine pancreas rough microsomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKd: 2.06E+4nMAssay Description:Binding affinity to human His-tagged HSP90alpha N-terminal domain (1 to 236 residues) expressed in Escherichia coli BL21star (DE3) by biolayer interf...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of FITC-geldanamycin binding to human His-tagged HSP90alpha N-terminal domain (1 to 236 residues) expressed in Escherichia coli BL21star (...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of FITC-geldanamycin binding to human His-tagged HSP90alpha N-terminal domain (1 to 236 residues) expressed in Escherichia coli BL21star (...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of FITC-geldanamycin binding to canine GRP94 incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of FITC-geldanamycin binding to canine GRP94 incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Binding affinity to GRP94 N-domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Binding affinity to GRP94 N-domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of human recombinant HSP90alpha expressed in Escherichia coli by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.92E+4nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of human recombinant HSP90alpha expressed in Escherichia coli by fluorescence polarization assayMore data for this Ligand-Target Pair
