Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50003224
TargetEphrin type-A receptor 2(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50468252(CHEMBL4281226)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to human EphA2 ligand binding domain (27 to 200 residues) expressed in Escherichia coli Rosetta-gami B(DE3) by ITCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 4(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM223300(EphA4-LBC inhibitor, Compound 22)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to EphA4 ligand binding domain (unknown origin) by ITCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50468253(CHEMBL4283329)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human EphA2 ligand binding domain (27 to 200 residues) expressed in Escherichia coli Rosetta-gami B(DE3) by ITCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Mouse)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50428234(CHEMBL2336575)
Affinity DataKd:  700nMAssay Description:Binding affinity to histidine-tagged mouse EphA2 Fc fusion protein by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50468254(CHEMBL4291811)
Affinity DataKd:  2nMAssay Description:Binding affinity to Fc-tagged EphB4 (unknown origin) assessed as reduction in ephrin-B2 binding by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50468255(CHEMBL4291184)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to human EphA2 ligand binding domain (27 to 200 residues) expressed in Escherichia coli Rosetta-gami B(DE3) by ITCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 4(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM223311(123C4)
Affinity DataKd:  420nMAssay Description:Binding affinity to EphA4 ligand binding domain (unknown origin) by ITCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50468256(CHEMBL4276804)
Affinity DataKd:  12nMAssay Description:Binding affinity to EphB2 (unknown origin) by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Mouse)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50468257(CHEMBL4227246)
Affinity DataKd:  700nMAssay Description:Binding affinity to histidine-tagged mouse EphA2 Fc fusion protein by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Mouse)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50236238(5beta-cholanic acid-3alpha-ol | CHEMBL1478 | (3alp...)
Affinity DataIC50: 5.70E+4nMAssay Description:Displacement of biotinylated ephrinA1-Fc from recombinant mouse EphA2 Fc chimera protein by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50234950(CHEMBL4059908)
Affinity DataKi: >1.50E+4nMAssay Description:Binding affinity to EphA2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed