BindingDB PrimarySearch

Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50005397

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50080337((R)-1-{2-[2,2-Bis-(3-methyl-thiophen-2-yl)-vinylox...)

IC50: 14nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491721(CHEMBL2387654)

IC50: 100nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50039251((R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)pi...)

IC50: 132nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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3D Structure (crystal)

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491707(CHEMBL2387677)

IC50: 302nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491713(CHEMBL2387675)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491722(CHEMBL2387655)

IC50: 339nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491705(CHEMBL2387667)

IC50: 398nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491709(CHEMBL2387671)

IC50: 631nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50020891((R)-1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carbo...)

IC50: 692nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491708(CHEMBL2387659)

IC50: 759nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491703(CHEMBL2387657)

IC50: 794nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491706(CHEMBL2387673)

IC50: 1.10E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491710(CHEMBL2387669)

IC50: 1.18E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491720(CHEMBL2387681)

IC50: 1.86E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491718(CHEMBL2387663)

IC50: 2.63E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491727(CHEMBL2387670)

IC50: 2.69E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491725(CHEMBL2387665)

IC50: 3.02E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491716(CHEMBL2387666)

IC50: 4.17E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491715(CHEMBL2387668)

IC50: 4.57E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491714(CHEMBL2387674)

IC50: 6.76E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491726(CHEMBL2387680)

IC50: 7.08E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)

IC50: 7.24E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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3D Structure (crystal)

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491723(CHEMBL2387661)

IC50: 7.59E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491717(CHEMBL2387664)

IC50: 8.13E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50003624((RS)-nipecotic acid | CHEMBL277498 | Nipecotic | P...)

IC50: 8.51E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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3D Structure (crystal)

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491702(CHEMBL2387672)

IC50: 8.91E+3nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491712(CHEMBL2387676)

IC50: 1.02E+4nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491711(CHEMBL2387658)

IC50: 1.07E+4nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)

IC50: 1.15E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491709(CHEMBL2387671)

IC50: 1.95E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50003624((RS)-nipecotic acid | CHEMBL277498 | Nipecotic | P...)

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491713(CHEMBL2387675)

IC50: 2.00E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491719(CHEMBL2387660)

IC50: 2.09E+4nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491724(CHEMBL2387679)

IC50: 2.51E+4nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)

IC50: 2.75E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491707(CHEMBL2387677)

IC50: 2.82E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 1(Rat)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491704(CHEMBL2387662)

IC50: 2.95E+4nMAssay Description:Inhibition of mouse GAT1 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491710(CHEMBL2387669)

IC50: 3.47E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491716(CHEMBL2387666)

IC50: 3.72E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491706(CHEMBL2387673)

IC50: 5.01E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491704(CHEMBL2387662)

IC50: 6.03E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491708(CHEMBL2387659)

IC50: 6.61E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491706(CHEMBL2387673)

IC50: 9.12E+4nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491711(CHEMBL2387658)

IC50: 1.41E+5nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50020891((R)-1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carbo...)

IC50: 1.95E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491704(CHEMBL2387662)

IC50: 3.39E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 3(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50491711(CHEMBL2387658)

IC50: 3.72E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50020891((R)-1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carbo...)

IC50: 3.72E+5nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Sodium- and chloride-dependent GABA transporter 2(Mouse)
Ludwig-Maximilians-University Munich

Curated by ChEMBL

BDBM50003624((RS)-nipecotic acid | CHEMBL277498 | Nipecotic | P...)

IC50: 5.25E+5nMAssay Description:Inhibition of mouse GAT2 expressed in HEK cells assessed as inhibition of [3H]-GABA uptake after 25 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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