Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50005974
TargetThromboxane-A synthase(Rat)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50017896(CHEMBL11662 | (E)-3-(4-Imidazol-1-ylmethyl-phenyl)...)
Affinity DataIC50: 200nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Rat)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50017896(CHEMBL11662 | (E)-3-(4-Imidazol-1-ylmethyl-phenyl)...)
Affinity DataIC50: 200nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50017896(CHEMBL11662 | (E)-3-(4-Imidazol-1-ylmethyl-phenyl)...)
Affinity DataIC50: 300nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Rat)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)
Affinity DataIC50: 300nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50017896(CHEMBL11662 | (E)-3-(4-Imidazol-1-ylmethyl-phenyl)...)
Affinity DataIC50: 300nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)
Affinity DataIC50: 500nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50017896(CHEMBL11662 | (E)-3-(4-Imidazol-1-ylmethyl-phenyl)...)
Affinity DataIC50: 900nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Rat)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)
Affinity DataIC50: 1.30E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)
Affinity DataIC50: 1.60E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)
Affinity DataIC50: 1.60E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Rat)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)
Affinity DataIC50: 1.70E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)
Affinity DataIC50: 2.30E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Rat)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)
Affinity DataIC50: 3.30E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)
Affinity DataIC50: 3.90E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)
Affinity DataIC50: 8.70E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed