Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50007072
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506026(CHEMBL4437206)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506037(CHEMBL4518406)
Affinity DataEC50:  0.0830nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506036(CHEMBL4443604)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506035(CHEMBL4437702)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506034(CHEMBL4444538)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506033(CHEMBL4473653)
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506032(CHEMBL4578949)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506031(CHEMBL4562873)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506030(CHEMBL4565753)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506029(CHEMBL4441946)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506028(CHEMBL4444303)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506027(CHEMBL4587131)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  0.0470nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506025(CHEMBL4454971)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506024(CHEMBL4461195)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506023(CHEMBL4525712)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506022(CHEMBL4561041)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506021(CHEMBL4526882)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  0.0930nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506020(CHEMBL4450702)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506019(CHEMBL4473347)
Affinity DataEC50:  0.0620nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  0.0620nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506019(CHEMBL4473347)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506017(CHEMBL4547328)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetApelin receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506016(CHEMBL4569052)
Affinity DataEC50:  7.40nMAssay Description:Agonist activity at human APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed