Compile Data Set for Download or QSAR
Report error Found 94 Enz. Inhib. hit(s) with all data for entry = 50007259
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060458((Z)-7-[(1R,2S,3S,4S)-3-(Naphthalene-2-sulfonylamin...)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060454((Z)-7-{(1R,2R,3S,5S)-2-[(5-Fluoro-benzo[b]thiophen...)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060462(CHEMBL116837 | S-5751 | (Z)-7-{(1R,2R,3S,5S)-2-[(5...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060462(CHEMBL116837 | S-5751 | (Z)-7-{(1R,2R,3S,5S)-2-[(5...)
Affinity DataIC50: 1nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060453((Z)-7-{(1R,2R,3S,5S)-2-[(6-Hydroxy-benzo[b]thiophe...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060454((Z)-7-{(1R,2R,3S,5S)-2-[(5-Fluoro-benzo[b]thiophen...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060453((Z)-7-{(1R,2R,3S,5S)-2-[(6-Hydroxy-benzo[b]thiophe...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060459((Z)-7-{(1R,2R,3S,5S)-2-[(Benzo[b]thiophene-7-carbo...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060465((Z)-7-[(1S,2R,3R,4R)-3-(4-Phenylethynyl-benzenesul...)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060452((Z)-7-{(1R,2R,3S,5S)-2-[(Benzo[b]thiophene-3-carbo...)
Affinity DataIC50: 22nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060459((Z)-7-{(1R,2R,3S,5S)-2-[(Benzo[b]thiophene-7-carbo...)
Affinity DataIC50: 26nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060463((Z)-7-[(1R,2R,6S,7R)-3-(4-Phenylazo-benzenesulfony...)
Affinity DataIC50: 27nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060447((Z)-7-[(1S,2R,3R,4R)-3-(2-Methoxy-dibenzofuran-3-s...)
Affinity DataIC50: 27nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060460((Z)-7-{(1R,2R,3S,5S)-6,6-Dimethyl-2-[(1H-pyrrole-2...)
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060452((Z)-7-{(1R,2R,3S,5S)-2-[(Benzo[b]thiophene-3-carbo...)
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060467((Z)-7-{(1R,2R,3S,5S)-2-[(Dibenzofuran-2-carbonyl)-...)
Affinity DataIC50: 32nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060455((Z)-7-{(1R,2R,3S,5S)-6,6-Dimethyl-2-[(thiophene-3-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060445((Z)-7-[(1R,2S,3S,4S)-3-(Biphenyl-4-sulfonylamino)-...)
Affinity DataIC50: 44nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((Z)-7-[(1S,2R,3R,4R)-3-(2-Phenyl-1H-indole-6-sulfo...)
Affinity DataIC50: 47nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060460((Z)-7-{(1R,2R,3S,5S)-6,6-Dimethyl-2-[(1H-pyrrole-2...)
Affinity DataIC50: 64nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060447((Z)-7-[(1S,2R,3R,4R)-3-(2-Methoxy-dibenzofuran-3-s...)
Affinity DataIC50: 68nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060461((Z)-7-[(1S,2R,3R,4R)-3-(Dibenzofuran-2-sulfonylami...)
Affinity DataIC50: 70nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060462(CHEMBL116837 | S-5751 | (Z)-7-{(1R,2R,3S,5S)-2-[(5...)
Affinity DataIC50: 96nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((Z)-7-[(1S,2R,3R,4R)-3-(2-Phenyl-1H-indole-6-sulfo...)
Affinity DataIC50: 120nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060461((Z)-7-[(1S,2R,3R,4R)-3-(Dibenzofuran-2-sulfonylami...)
Affinity DataIC50: 130nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060466(7-[6,6-Dimethyl-2-(4-phenylazo-benzoylamino)-bicyc...)
Affinity DataIC50: 150nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060459((Z)-7-{(1R,2R,3S,5S)-2-[(Benzo[b]thiophene-7-carbo...)
Affinity DataIC50: 210nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060467((Z)-7-{(1R,2R,3S,5S)-2-[(Dibenzofuran-2-carbonyl)-...)
Affinity DataIC50: 220nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060468((Z)-7-[(1R,2R,3S,5S)-2-(Dibenzofuran-2-sulfonylami...)
Affinity DataIC50: 240nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060465((Z)-7-[(1S,2R,3R,4R)-3-(4-Phenylethynyl-benzenesul...)
Affinity DataIC50: 250nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060451((Z)-7-[(1S,2R,3R,4R)-3-(7-Nitro-dibenzofuran-2-sul...)
Affinity DataIC50: 250nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060467((Z)-7-{(1R,2R,3S,5S)-2-[(Dibenzofuran-2-carbonyl)-...)
Affinity DataIC50: 270nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060465((Z)-7-[(1S,2R,3R,4R)-3-(4-Phenylethynyl-benzenesul...)
Affinity DataIC50: 280nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060463((Z)-7-[(1R,2R,6S,7R)-3-(4-Phenylazo-benzenesulfony...)
Affinity DataIC50: 320nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060446(7-(2-Benzoylamino-6,6-dimethyl-bicyclo[3.1.1]hept-...)
Affinity DataIC50: 360nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060452((Z)-7-{(1R,2R,3S,5S)-2-[(Benzo[b]thiophene-3-carbo...)
Affinity DataIC50: 380nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060466(7-[6,6-Dimethyl-2-(4-phenylazo-benzoylamino)-bicyc...)
Affinity DataIC50: 380nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060453((Z)-7-{(1R,2R,3S,5S)-2-[(6-Hydroxy-benzo[b]thiophe...)
Affinity DataIC50: 410nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060457((Z)-7-[(1S,2R,3R,4R)-3-(Naphthalene-2-sulfonylamin...)
Affinity DataIC50: 420nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060454((Z)-7-{(1R,2R,3S,5S)-2-[(5-Fluoro-benzo[b]thiophen...)
Affinity DataIC50: 430nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060464((+) 7-[3-(Biphenyl-4-sulfonylamino)-bicyclo[2.2.1]...)
Affinity DataIC50: 450nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060445((Z)-7-[(1R,2S,3S,4S)-3-(Biphenyl-4-sulfonylamino)-...)
Affinity DataIC50: 460nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060445((Z)-7-[(1R,2S,3S,4S)-3-(Biphenyl-4-sulfonylamino)-...)
Affinity DataIC50: 520nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060466(7-[6,6-Dimethyl-2-(4-phenylazo-benzoylamino)-bicyc...)
Affinity DataIC50: 540nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060464((+) 7-[3-(Biphenyl-4-sulfonylamino)-bicyclo[2.2.1]...)
Affinity DataIC50: 600nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060457((Z)-7-[(1S,2R,3R,4R)-3-(Naphthalene-2-sulfonylamin...)
Affinity DataIC50: 670nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060456((+) 7-[3-(4-Phenoxy-benzenesulfonylamino)-bicyclo[...)
Affinity DataIC50: 720nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane A2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060449(7-[6,6-Dimethyl-2-(4-phenylazo-benzenesulfonylamin...)
Affinity DataIC50: 740nMAssay Description:Inhibition of [3H]- (+)-S-145 specific binding to human platelet membranes in TXA2 receptor (TP) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060456((+) 7-[3-(4-Phenoxy-benzenesulfonylamino)-bicyclo[...)
Affinity DataIC50: 780nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060468((Z)-7-[(1R,2R,3S,5S)-2-(Dibenzofuran-2-sulfonylami...)
Affinity DataIC50: 780nMAssay Description:Inhibition of [3H]PGD-2 specific binding to Prostaglandin D2 receptor from human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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