Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50007883
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50068974(CGP-57698 | 2,2-Diethyl-N-[3-(7-fluoro-quinolin-2-...)
Affinity DataIC50: 0.200nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215369(CHEMBL368290)
Affinity DataIC50: 0.300nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215411(CHEMBL425675)
Affinity DataIC50: 0.400nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215410(CHEMBL369421)
Affinity DataIC50: 0.5nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50068987(N-[3-(7-Chloro-quinolin-2-ylmethoxy)-phenyl]-2,2-d...)
Affinity DataIC50: 0.800nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50068980(2,2-Diethyl-N-[3-(quinolin-2-ylmethoxy)-phenyl]-su...)
Affinity DataIC50: 0.900nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215370(CHEMBL174265)
Affinity DataIC50: 1nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215372(CHEMBL175419)
Affinity DataIC50: 1.40nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215394(CHEMBL368666)
Affinity DataIC50: 2nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215399(CHEMBL174575)
Affinity DataIC50: 2nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215397(CHEMBL173523)
Affinity DataIC50: 3nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215371(CHEMBL174743)
Affinity DataIC50: 4nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215390(CHEMBL176961)
Affinity DataIC50: 4nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50009073(cyclopentyl 3-(2-methoxy-4-((o-tolylsulfonyl)carba...)
Affinity DataIC50: 5nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215353(CHEMBL177814)
Affinity DataIC50: 6nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50068974(CGP-57698 | 2,2-Diethyl-N-[3-(7-fluoro-quinolin-2-...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215407(CHEMBL175382)
Affinity DataIC50: 6.40nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215376(CHEMBL362228)
Affinity DataIC50: 7.30nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50068980(2,2-Diethyl-N-[3-(quinolin-2-ylmethoxy)-phenyl]-su...)
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215398(CHEMBL174687)
Affinity DataIC50: 9nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215396(CHEMBL176654)
Affinity DataIC50: 9nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215373(CHEMBL178049)
Affinity DataIC50: 10nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215355(CHEMBL368001)
Affinity DataIC50: 11nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215412(CHEMBL177172)
Affinity DataIC50: 11nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215409(CHEMBL174440)
Affinity DataIC50: 24nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50009073(cyclopentyl 3-(2-methoxy-4-((o-tolylsulfonyl)carba...)
Affinity DataIC50: 44nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50068987(N-[3-(7-Chloro-quinolin-2-ylmethoxy)-phenyl]-2,2-d...)
Affinity DataIC50: 64nMAssay Description:In vitro inhibition of [3H]LTD4 binding to guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215374(CHEMBL426941)
Affinity DataIC50: 80nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215408(CHEMBL176412)
Affinity DataIC50: 140nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215354(CHEMBL174655)
Affinity DataIC50: 200nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215395(CHEMBL174544)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50215375(CHEMBL174645)
Affinity DataIC50: 3.90E+3nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed