Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50010095
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50240586(CHEMBL4098982)
Affinity DataIC50: 91nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50535120(CHEMBL4451097)
Affinity DataIC50: 370nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50535123(CHEMBL4552544)
Affinity DataIC50: 1.09E+3nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM36363(CID6851947 | PAC-1 | US10166229, Example PAC-1)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50535119(CHEMBL4457255)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50535121(CHEMBL4452014)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Istituto Di Scienze E Tecnologie Molecolari (Istm)

Curated by ChEMBL
LigandPNGBDBM50535122(CHEMBL4452878)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed