Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50011226
TargetHistone acetyltransferase p300(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataKd:  3.18E+7nMAssay Description:Reverse ITC (compound as receptor). Domain start/stop: A1040-S1171More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 66nMAssay Description:Alphascreen assay. Binding to CREBBPA (domain start/stop: R1081-G1197) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 68nMAssay Description:Alphascreen assay. Binding to CREBBPA (domain start/stop: R1081-G1197) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 7.12E+3nMAssay Description:Alphascreen assay. Binding to BRD4A (domain start/stop: N44-E168) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 2.78E+4nMAssay Description:Alphascreen assay. Binding to BRD4A (domain start/stop: N44-E168) by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)