Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50012590
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120763(Cyclopentanecarboxylic acid (7-ethyl-2-phenyl-imid...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120761(Cyclopentanecarboxylic acid (7-methyl-2-phenyl-imi...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120767(Cyclopentanecarboxylic acid (7-isopropyl-2-phenyl-...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120759(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  11.8nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120765(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120764(Cyclopentanecarboxylic acid (2,7-diphenyl-imidazo[...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120767(Cyclopentanecarboxylic acid (7-isopropyl-2-phenyl-...)
Affinity DataKi:  17.4nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120763(Cyclopentanecarboxylic acid (7-ethyl-2-phenyl-imid...)
Affinity DataKi:  20.2nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120766(N-(2,7-Diphenyl-imidazo[1,2-a][1,3,5]triazin-4-yl)...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120759(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  27.2nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120766(N-(2,7-Diphenyl-imidazo[1,2-a][1,3,5]triazin-4-yl)...)
Affinity DataKi:  40nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120758(Cyclopentyl-(7-methyl-2-phenyl-imidazo[1,2-a][1,3,...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120760(Cyclohexanecarboxylic acid (7-methyl-2-phenyl-imid...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120760(Cyclohexanecarboxylic acid (7-methyl-2-phenyl-imid...)
Affinity DataKi:  202nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120754(Cyclohexylmethyl-(7-methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120753(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  231nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120757(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4-y...)
Affinity DataKi:  332nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120761(Cyclopentanecarboxylic acid (7-methyl-2-phenyl-imi...)
Affinity DataKi:  410nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120770(Adamantan-1-yl-(7-methyl-2-phenyl-imidazo[1,2-a][1...)
Affinity DataKi:  511nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120770(Adamantan-1-yl-(7-methyl-2-phenyl-imidazo[1,2-a][1...)
Affinity DataKi:  526nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120757(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4-y...)
Affinity DataKi:  682nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120753(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi:  855nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120764(Cyclopentanecarboxylic acid (2,7-diphenyl-imidazo[...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120757(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4-y...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120754(Cyclohexylmethyl-(7-methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120758(Cyclopentyl-(7-methyl-2-phenyl-imidazo[1,2-a][1,3,...)
Affinity DataKi:  2.25E+3nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120768(1-(7-Isopropyl-2-phenyl-imidazo[1,2-a][1,3,5]triaz...)
Affinity DataKi:  2.36E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120764(Cyclopentanecarboxylic acid (2,7-diphenyl-imidazo[...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120763(Cyclopentanecarboxylic acid (7-ethyl-2-phenyl-imid...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120768(1-(7-Isopropyl-2-phenyl-imidazo[1,2-a][1,3,5]triaz...)
Affinity DataKi:  3.05E+3nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120766(N-(2,7-Diphenyl-imidazo[1,2-a][1,3,5]triazin-4-yl)...)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120769(Benzyl-(7-methyl-2-phenyl-imidazo[1,2-a][1,3,5]tri...)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120758(Cyclopentyl-(7-methyl-2-phenyl-imidazo[1,2-a][1,3,...)
Affinity DataKi:  4.10E+3nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120761(Cyclopentanecarboxylic acid (7-methyl-2-phenyl-imi...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120762(1-(2,7-Diphenyl-imidazo[1,2-a][1,3,5]triazin-4-yla...)
Affinity DataKi:  5.80E+3nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120770(Adamantan-1-yl-(7-methyl-2-phenyl-imidazo[1,2-a][1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120753(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120754(Cyclohexylmethyl-(7-methyl-2-phenyl-imidazo[1,2-a]...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120755(1-(7-Ethyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120755(1-(7-Ethyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-4...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120756(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120762(1-(2,7-Diphenyl-imidazo[1,2-a][1,3,5]triazin-4-yla...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50120756(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor in bovine cortical membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120769(Benzyl-(7-methyl-2-phenyl-imidazo[1,2-a][1,3,5]tri...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120767(Cyclopentanecarboxylic acid (7-isopropyl-2-phenyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120760(Cyclohexanecarboxylic acid (7-methyl-2-phenyl-imid...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120759(N-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120768(1-(7-Isopropyl-2-phenyl-imidazo[1,2-a][1,3,5]triaz...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- CGS-21680 from Adenosine A2a receptor in bovine striatal membranes.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120765(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50120756(1-(7-Methyl-2-phenyl-imidazo[1,2-a][1,3,5]triazin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]AB-MECA from Adenosine A3 receptor in bovine cortical membranes in the presence of 20 nM DPCPX.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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