Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50014037
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572018(CHEMBL4854351)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572021(CHEMBL4864112)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572019(CHEMBL4855879)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50010586(CHEMBL70565 | (-)-1-Propyl-2,3,10,10a-tetrahydro-1...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572022(CHEMBL4875181)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572025(CHEMBL4852472)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572004(CHEMBL4863032)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572007(CHEMBL4862320)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572014(CHEMBL4853503)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572024(CHEMBL4862790)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi: <10nMAssay Description:Partial agonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572005(CHEMBL4875008)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572008(CHEMBL4848907)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572016(CHEMBL4860687)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572010(CHEMBL4849734)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572020(CHEMBL4864813)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572027(CHEMBL4848710)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572001(CHEMBL4845838)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572000(CHEMBL4878501)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572002(CHEMBL4862399)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572015(CHEMBL4864074)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50571999(CHEMBL4878826)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572012(CHEMBL4855711)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572028(CHEMBL4864969)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572017(CHEMBL4877715)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572006(CHEMBL4878577)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572026(CHEMBL4853993)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572009(CHEMBL4869122)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572023(CHEMBL4862275)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50010586(CHEMBL70565 | (-)-1-Propyl-2,3,10,10a-tetrahydro-1...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572003(CHEMBL4854126)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572013(CHEMBL4869668)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(3) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572011(CHEMBL4848199)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572012(CHEMBL4855711)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50571999(CHEMBL4878826)
Affinity DataKi:  473nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572002(CHEMBL4862399)
Affinity DataKi:  563nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572027(CHEMBL4848710)
Affinity DataKi:  568nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572007(CHEMBL4862320)
Affinity DataKi:  568nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572020(CHEMBL4864813)
Affinity DataKi:  589nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572028(CHEMBL4864969)
Affinity DataKi:  642nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572006(CHEMBL4878577)
Affinity DataKi:  663nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572023(CHEMBL4862275)
Affinity DataKi:  688nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572021(CHEMBL4864112)
Affinity DataKi:  697nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572004(CHEMBL4863032)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572000(CHEMBL4878501)
Affinity DataKi:  723nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572013(CHEMBL4869668)
Affinity DataKi:  728nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572018(CHEMBL4854351)
Affinity DataKi:  732nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetD(2) dopamine receptor(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50572024(CHEMBL4862790)
Affinity DataKi:  744nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 68 total ) | Next | Last >>
Jump to: